SCHEMBL20143957

SCHEMBL20143957

CCc1cnc(C#N)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.43
NAAA Q02083 1/20 0.39
CTSS P25774 2/20 0.35
CTSK P43235 2/20 0.35
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HPGD P15428 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM4E B2RXH2 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MAPT P10636 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PANK3 Q9H999 1/20 0.32
EGLN2 Q96KS0 1/20 0.32
PARP1 P09874 1/20 0.31
CRHBP P24387 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19187070 0.80 CYP2A6 (0.48) CYP2A6NAAACTSSCTSKTSHR
SCHEMBL9455422 0.76 NAAA (0.39) NAAACTSSEGLN2
SCHEMBL19971709 0.76 NAAA (0.39) NAAAEGLN2
SCHEMBL24078807 0.76 L3MBTL1 (0.33) TDP1KDM4EL3MBTL1SMN1; SMN2NOS3
SCHEMBL6476454 0.76 LOXL2 (0.43) NAAAKDM4EL3MBTL1EGLN2ALDH1A1
SCHEMBL24149399 0.76 NAAA (0.39) NAAATDP1KDM4EL3MBTL1MAPT
SCHEMBL15858738 0.76 CTSS (0.38) NAAACTSSCTSKPANK3
SCHEMBL15858740 0.76 CTSK (0.37) NAAACTSSCTSK
SCHEMBL17778285 0.74 NAAA (0.45) NAAACTSSCTSKHPGDEGLN2
Hydrochloric Acid SCHEMBL6476958 0.74 LOXL2 (0.41) NAAAKDM4EL3MBTL1EGLN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230250129-A1 NEUROACTIVE STEROIDS AND COMPOSITIONS THEREOF SAGE THERAPEUTICS, INC. 2023-08-10 US disclosed
WO-2023134629-A1 NUCLEAR TRANSPORT REGULATOR AND USE THEREOF 上海海雁医药科技有限公司 2023-07-20 WO disclosed
US-20220020935-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES Beijing Summer Sprout Technology Co., Ltd. (CN) 2022-01-20 US disclosed
US-20210087147-A1 SELECTIVE INHIBITORS OF NLRP3 INFLAMMASOME NodThera Limited (GB) 2021-03-25 US disclosed
EP-3541810-B1 TRIAZOLE PHENYL COMPOUNDS AS AGONISTS OF THE APJ RECEPTOR AMGEN INC (US) 2020-12-23 EP disclosed
US-9969694-B2 N-(arylalkyl)-N′-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors ARRAY BIOPHARMA INC. (US) 2018-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230250129-A1 NEUROACTIVE STEROIDS AND COMPOSITIONS THEREOF MC2R, NR3C2, AVPR1B CYP2A6 349/4885NAAA 937/4885CTSS 2518/4885
US-20210087147-A1 SELECTIVE INHIBITORS OF NLRP3 INFLAMMASOME NLRP3, NOD1, NLRP1 CYP2A6 3770/4885NAAA 3454/4885CTSS 941/4885
US-20220020935-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD1, OCIAD2, LEF1 CYP2A6 4351/4885NAAA 4627/4885CTSS 1036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.