SCHEMBL202283

SCHEMBL202283

C#CC(O)(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
USP2 O75604 1/20 0.43
CYP19A1 P11511 4/20 0.41
KCNN4 O15554 6/20 0.40
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
HSD11B1 P28845 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
HTT P42858 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
XBP1 P17861 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KCNE1 P15382 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217833 0.92 KCNN4 (0.47) RAB9AUSP2CYP19A1KCNN4CYP3A4
SCHEMBL4041575 0.90 KCNN4 (0.38) RAB9AUSP2CYP19A1KCNN4CYP3A4
SCHEMBL11479898 0.87 KCNN4 (0.43) RAB9AUSP2KCNN4CYP3A4CYP2D6
SCHEMBL3143169 0.85 NFE2L2 (0.46) RAB9AHSD11B1KMT2ANPC1SMN1; SMN2
SCHEMBL11485302 0.82 KCNN4 (0.40) KCNN4KCNE1KCNQ1L3MBTL1LMNA
SCHEMBL1817358 0.80 SMN1; SMN2 (0.45) CYP3A4CYP2D6CYP2C19SMN1; SMN2GAA
SCHEMBL1958061 0.80 NPC1 (0.53) RAB9AUSP2HSD11B1HTTKMT2A
SCHEMBL1962637 0.79 AKR1C3 (0.49) USP2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1959801 0.79 FAAH (0.47) CYP2D6CYP2C19SMN1; SMN2L3MBTL1LMNA
SCHEMBL10049978 0.78 ESR1 (0.44) RAB9ACYP3A4KMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113227099-B Articles comprising indolonaphthopyrans 光学转变有限公司 2025-03-11 CN disclosed
US-12247035-B2 Articles comprising indolenaphthopyrans TRANSITIONS OPTICAL, LTD. (IE) 2025-03-11 US disclosed
EP-3898635-B1 ARTICLES COMPRISING INDOLONAPHTHOPYRANS TRANSITIONS OPTICAL LTD (IE) 2024-12-04 EP disclosed
US-11897894-B2 Indolenaphthopyrans TRANSITIONS OPTICAL, LTD. (IE) 2024-02-13 US disclosed
EP-3268375-B1 PHOTOCHROMIC THIENOCHROMENE COMPOUNDS TRANSITIONS OPTICAL INC (US) 2022-06-15 EP disclosed
CN-107253943-B Photochromic compounds and compositions 光学转变公司 2022-05-17 CN disclosed
US-20220064175-A1 Articles Comprising Indolenaphthopyrans TRANSITIONS OPTICAL, LTD. (IE) 2022-03-03 US disclosed
EP-3898844-A1 INDOLENAPHTHOPYRANS AND PHOTOCHROMIC COMPOSITIONS COMPRISING THEM Transitions Optical, Ltd. (IE) 2021-10-27 EP disclosed
EP-3898635-A1 ARTICLES COMPRISING INDOLENAPHTHOPYRANS Transitions Optical, Ltd. (IE) 2021-10-27 EP disclosed
US-20210317129-A1 Indolenaphthopyrans TRANSITIONS OPTICAL, LTD. (IE) 2021-10-14 US disclosed
EP-2401269-A1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2012-01-04 EP disclosed
US-20110143141-A1 Photochromic compounds and compositions TRANSITIONS OPTICAL, INC. (US) 2011-06-16 US disclosed
US-20110129678-A1 Photochromic compounds and compositions TRANSITIONS OPTICAL, INC. (US) 2011-06-02 US disclosed
US-20100234415-A1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LLC 2010-09-16 US disclosed
WO-2010099039-A1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-09-02 WO disclosed
EP-1963896-B1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL INC (US) 2010-02-10 EP disclosed
US-7556751-B2 Photochromic materials having electron-withdrawing substituents TRANSITIONS OPTICAL, INC. (US) 2009-07-07 US disclosed
EP-1963896-A1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL, INC. (US) 2008-09-03 EP disclosed
WO-2007073462-A1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL, INC. (US) 2007-06-28 WO disclosed
US-20070138449-A1 Photochromic materials having electron-withdrawing substituents TRANSITIONS OPTICAL LIMITED (IE) 2007-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110143141-A1 Photochromic compounds and compositions CCNA1, CRY1, CCNT1 RAB9A 1829/4885USP2 3531/4885CYP19A1 138/4885
US-20210317129-A1 Indolenaphthopyrans AHR, TDO2, TPH2 RAB9A 2996/4885USP2 2952/4885CYP19A1 966/4885
US-11897894-B2 Indolenaphthopyrans AHR, TDO2, TPH2 RAB9A 2996/4885USP2 2952/4885CYP19A1 966/4885
US-20100234415-A1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS PTGER2, PTGDR2, PTGDR RAB9A 3377/4885USP2 2639/4885CYP19A1 875/4885
US-20220064175-A1 Articles Comprising Indolenaphthopyrans CDC25B, ACTB, CCNB1 RAB9A 1667/4885USP2 1455/4885CYP19A1 2214/4885
US-20110129678-A1 Photochromic compounds and compositions CRY2, CRY1, PPOX RAB9A 2888/4885USP2 3017/4885CYP19A1 1449/4885
US-12247035-B2 Articles comprising indolenaphthopyrans ACTB, CCNB1, HMBS RAB9A 2299/4885USP2 1222/4885CYP19A1 2119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.