SCHEMBL20527221

SCHEMBL20527221

Cn1cc(Br)nc1C(=O)Nc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.47
POLB P06746 1/20 0.46
BACE1 P56817 2/20 0.45
RAB9A P51151 7/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
NPC1 O15118 4/20 0.43
TSHR P16473 1/20 0.43
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
RECQL P46063 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALOX15 P16050 1/20 0.42
CDK2 P24941 1/20 0.42
NAMPT P43490 1/20 0.42
HTT P42858 1/20 0.41
HPGD P15428 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16693604 0.83 RAB9A (0.50) POLBBACE1RAB9AMEN1KMT2A
SCHEMBL20086628 0.82 POLB (0.46) ATRPOLBRAB9AMEN1KMT2A
SCHEMBL16691855 0.79 SMN1; SMN2 (0.47) ATRPOLBRAB9AMEN1KMT2A
SCHEMBL20833871 0.78 HPGD (0.55) POLBMEN1KMT2AHDAC2HDAC8
SCHEMBL20527174 0.76 SMN1; SMN2 (0.50) ATRPOLBRAB9AMEN1KMT2A
SCHEMBL21316476 0.73 NAMPT (0.46) POLBRAB9AMEN1KMT2ANPC1
SCHEMBL14583507 0.72 NAMPT (0.74) ATRPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL14156000 0.71 BACE1 (0.33) POLBBACE1HDAC8L3MBTL1SMN1; SMN2
SCHEMBL25732873 0.71 BCAT2 (0.48) ATRPOLBRAB9AMEN1KMT2A
SCHEMBL21451631 0.70 NAMPT (0.47) RAB9ANPC1TSHRSMN1; SMN2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12583857-B2 Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines PHEON THERAPEUTICS LTD (GB) 2026-03-24 US disclosed
US-20250011317-A1 ANTI-PROLIFERATIVE AGENTS PHEON THERAPEUTICS LTD (GB) 2025-01-09 US disclosed
US-11912700-B2 Anti-proliferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines PHEON THERAPEUTICS LTD (GB) 2024-02-27 US disclosed
US-11912700-B2 Anti-proliferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines PHEON THERAPEUTICS LTD (GB) 2024-02-27 US disclosed
US-11912700-B2 Anti-proliferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines PHEON THERAPEUTICS LTD (GB) 2024-02-27 US disclosed
US-20230302142-A1 Cytotoxic Agents Pheon Therapeutics Ltd. (GB) 2023-09-28 US disclosed
US-20230302142-A1 Cytotoxic Agents Pheon Therapeutics Ltd. (GB) 2023-09-28 US disclosed
US-20230302142-A1 Cytotoxic Agents Pheon Therapeutics Ltd. (GB) 2023-09-28 US disclosed
EP-4188927-A1 CYTOTOXIC AGENTS Pheon Therapeutics Ltd (GB) 2023-06-07 EP disclosed
WO-2022023735-A1 CYTOTOXIC AGENTS FEMTOGENIX LIMITED (GB) 2022-02-03 WO disclosed
US-20210206763-A1 Anti-Proliferative Agents PHEON THERAPEUTICS LTD (GB) 2021-07-08 US disclosed
US-20210206763-A1 Anti-Proliferative Agents PHEON THERAPEUTICS LTD (GB) 2021-07-08 US disclosed
US-10975072-B2 Substituted 6a,7,8,9,10,12-hexahydrobenzo[e]pyrido[1,2-a][1,4]diazepines as anti-proliferative agents FEMTOGENIX LIMITED 2021-04-13 US disclosed
US-10975072-B2 Substituted 6a,7,8,9,10,12-hexahydrobenzo[e]pyrido[1,2-a][1,4]diazepines as anti-proliferative agents FEMTOGENIX LIMITED 2021-04-13 US disclosed
US-10975074-B2 Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines FEMTOGENIX LIMITED 2021-04-13 US disclosed
US-10975074-B2 Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines FEMTOGENIX LIMITED 2021-04-13 US disclosed
US-20190308970-A1 ANTI-LIFERATIVE AGENTS COMPRISING SUBSTITUTED PYRROLO-, INDOLINO- OR TETRAHYDROISOQUINOLINE-BENZODIAZEPINES PHEON THERAPEUTICS LTD (GB) 2019-10-10 US disclosed
US-20190308970-A1 ANTI-LIFERATIVE AGENTS COMPRISING SUBSTITUTED PYRROLO-, INDOLINO- OR TETRAHYDROISOQUINOLINE-BENZODIAZEPINES PHEON THERAPEUTICS LTD (GB) 2019-10-10 US disclosed
US-20180339985-A1 PDD COMPOUNDS FEMTOGENIX LIMITED (GB) 2018-11-29 US disclosed
US-20180291021-A1 PDD COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2018-10-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210206763-A1 Anti-Proliferative Agents CCND2, BRD2, DRD2 ATR 2973/4885POLB 127/4885BACE1 4262/4885
US-10975074-B2 Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines CNR1, GABRA1, BAK1 ATR 1522/4885POLB 307/4885BACE1 2260/4885
US-12583857-B2 Anti-liferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines CNR1, MTNR1B, MTNR1A ATR 3640/4885POLB 2395/4885BACE1 1861/4885
US-20250011317-A1 ANTI-PROLIFERATIVE AGENTS CCND2, BRD2, CCND3 ATR 2147/4885POLB 104/4885BACE1 4527/4885
US-10975072-B2 Substituted 6a,7,8,9,10,12-hexahydrobenzo[e]pyrido[1,2-a][1,4]diazepines as anti-proliferative agents PDCD1, CCND1, PDCD6 ATR 3396/4885POLB 876/4885BACE1 3277/4885
US-20190308970-A1 ANTI-LIFERATIVE AGENTS COMPRISING SUBSTITUTED PYRROLO-, INDOLINO- OR TETRAHYDROISOQUINOLINE-BENZODIAZEPINES GABRA1, GABBR1, GABRA2 ATR 791/4885POLB 382/4885BACE1 3080/4885
US-20180291021-A1 PDD COMPOUNDS DRD1, DRD3, DRD2 ATR 3162/4885POLB 1536/4885BACE1 2908/4885
US-20230302142-A1 Cytotoxic Agents ANXA11, ANXA5, HAX1 ATR 1948/4885POLB 1962/4885BACE1 276/4885
US-11912700-B2 Anti-proliferative agents comprising substituted benzo[e]pyrido[1,2-a][1,4]diazepines MKI67, CCND2, CCND1 ATR 1760/4885POLB 231/4885BACE1 2243/4885
US-20180339985-A1 PDD COMPOUNDS DRD1, DRD3, DRD2 ATR 3433/4885POLB 1301/4885BACE1 2642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.