SCHEMBL21048922

SCHEMBL21048922

CCS(=O)(=O)Nc1ncc(C)cc1CNC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SETDB1 Q15047 1/20 0.34
PTPN1 P18031 2/20 0.34
PTPN2 P17706 1/20 0.34
F2 P00734 2/20 0.34
PRSS1 P07477 1/20 0.34
HPGD P15428 4/20 0.33
CYP2C9 P11712 3/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
NAMPT P43490 2/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
SLC13A5 Q86YT5 1/20 0.33
LMNA P02545 1/20 0.33
ESRRA P11474 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21048871 0.91 KDM4E (0.39) NPC1RAB9AHPGDKDM4EALDH1A1
SCHEMBL1230894 0.78 CYP2C9 (0.44) NPC1RAB9AF2HPGDCYP2C9
SCHEMBL21048873 0.72 JAK2 (0.46) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL21048923 0.71 PTK2 (0.49) ALDH1A1LMNA
SCHEMBL21048818 0.70 MMP1 (0.42) NPC1RAB9AALDH1A1MAPTMAPK1
SCHEMBL18595669 0.66 BRD4 (0.44) HPGDCYP2C9KDM4EALDH1A1GAA
SCHEMBL20483300 0.66 ADORA2A (0.46) NPC1RAB9AGAAMAPTLMNA
SCHEMBL15145602 0.66 MTNR1A (0.45) CYP2C9
SCHEMBL15343468 0.64 ADORA3 (0.41) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL18595670 0.64 PSIP1 (0.45) HPGDCYP2C9KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed