SCHEMBL21484847

SCHEMBL21484847

C[Si](C)(C)C#Cc1ccc(C(=O)CBr)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 12/20 0.56
PTPN1 P18031 6/20 0.48
MMP2 P08253 2/20 0.38
MMP12 P39900 2/20 0.38
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2321185 0.84 SMN1; SMN2 (0.46) GSK3BMMP2MMP12
SCHEMBL19707734 0.81 GSK3B (0.60) GSK3BPTPN1
SCHEMBL8049735 0.80 ALDH1A1 (0.43) RARBRARG
SCHEMBL9636621 0.78 HPGD (0.47) RARBRARG
SCHEMBL6036758 0.78 RARB (0.55) RARBRARG
SCHEMBL25093690 0.77 NOS1 (0.44) RARBRARG
SCHEMBL28655847 0.75 MMP2 (0.34) MMP2MMP12RARBRARG
SCHEMBL2321549 0.75 GSK3B (0.42) GSK3BMMP2MMP12RARBRARG
SCHEMBL1306384 0.74 GABRA1 (0.38)
SCHEMBL205280 0.74 GSK3B (0.80) GSK3BPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11584742-B2 Substituted aminothiazoles as inhibitors of nucleases MASARYKOVA UNIVERZITA (CZ) 2023-02-21 US disclosed
US-20220002282-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2022-01-06 US disclosed
EP-3556755-B1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES UNIV MASARYKOVA (CZ) 2021-11-17 EP disclosed
CN-112313229-A Substituted aminothiazoles as inhibitors of nucleases 马萨里克大学 2021-02-02 CN disclosed
EP-3556755-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES Masarykova univerzita (CZ) 2019-10-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11584742-B2 Substituted aminothiazoles as inhibitors of nucleases RNASEH1, DNASE1, FEN1 GSK3B 3281/4885PTPN1 3966/4885MMP2 993/4885
US-20220002282-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES RNASEH1, DNASE1, FEN1 GSK3B 3281/4885PTPN1 3966/4885MMP2 993/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.