SCHEMBL2170255

SCHEMBL2170255

NC(=O)C(Cc1ccc(Oc2ccc(F)cc2)cc1)NC(=O)CN1CCN(c2ccccn2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.57
MAPT P10636 2/20 0.57
TSHR P16473 2/20 0.57
GAA P10253 1/20 0.57
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
KDM4E B2RXH2 1/20 0.55
POLB P06746 1/20 0.50
DRD2 P14416 3/20 0.49
DRD3 P35462 3/20 0.49
DRD4 P21917 3/20 0.49
LMNA P02545 2/20 0.48
THRB P10828 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MMP1 P03956 1/20 0.48
MMP3 P08254 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2354704 0.90 ALDH1A1 (0.50) ALDH1A1MAPTTSHRGAAKDM4E
SCHEMBL2170811 0.86 MAPT (0.54) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL2170108 0.85 LMNA (0.52) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL2170332 0.85 ALDH1A1 (0.53) ALDH1A1MAPTTSHRMEN1KMT2A
SCHEMBL2350984 0.84 TRPA1 (0.44) ALDH1A1GAANPSR1HSD17B10SCN9A
SCHEMBL2171096 0.83 SCN9A (0.51) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL2169959 0.82 TSHR (0.58) ALDH1A1MAPTTSHRGAAMEN1
SCHEMBL2171705 0.81 MEN1 (0.60) ALDH1A1MAPTTSHRMEN1KMT2A
SCHEMBL2169958 0.81 SCN9A (0.47) ALDH1A1MEN1KMT2ALMNACA1
SCHEMBL2169808 0.80 SCN9A (0.48) ALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed