Water

Water

SCHEMBL21878445

O.O=C(O)c1ccc(-c2ccc(C(=O)O)c(C(=O)O)c2)cc1.O=C(O)c1ccc(-c2ccc(C(=O)O)c(C(=O)O)c2)cc1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR known ✓ P00374 1/20 0.50
GRIK1 known ✓ P39086 1/20 0.49
GRIK2 known ✓ Q13002 1/20 0.49
GRIK3 known ✓ Q13003 1/20 0.49
EGFR known ✓ P00533 1/20 0.48
BCL2L1 Q07817 1/20 0.52
BAD Q92934 1/20 0.52
RXRA P19793 3/20 0.52
RXRB P28702 3/20 0.52
KDM4E B2RXH2 3/20 0.52
HSD17B10 Q99714 2/20 0.52
LMNA P02545 1/20 0.52
HNF4A P41235 2/20 0.50
ACMSD Q8TDX5 2/20 0.50
CDC25B P30305 2/20 0.50
MCL1 Q07820 1/20 0.50
CDC25A P30304 1/20 0.50
ATM Q13315 1/20 0.50
GFER P55789 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29368917 0.98 BCL2L1 (0.54) BCL2L1BADRXRARXRBKDM4E
SCHEMBL6866233 0.98 BCL2L1 (0.54) BCL2L1BADRXRARXRBKDM4E
SCHEMBL16166057 0.90 ACMSD (0.61) RXRARXRBHSD17B10HNF4AACMSD
SCHEMBL28222622 0.89 KDM4E (0.60) KDM4EHSD17B10HNF4AACMSDCDC25B
Water SCHEMBL4330613 0.89 KMT2A (0.60) KDM4EHSD17B10HNF4AACMSDCDC25B
SCHEMBL29436303 0.89 KMT2A (0.60) KDM4EHSD17B10HNF4AACMSDCDC25B
SCHEMBL710222 0.89 KMT2A (0.60) KDM4EHSD17B10HNF4AACMSDCDC25B
SCHEMBL9550353 0.89 KMT2A (0.60) KDM4EHSD17B10HNF4AACMSDCDC25B
SCHEMBL9550390 0.88 POLB (0.63) KDM4EHSD17B10LMNAHNF4AACMSD
SCHEMBL30690398 0.87 KMT2A (0.62) KDM4EHSD17B10HNF4AACMSDCDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110799559-B Resin, resin composition, nonwoven fabric, fiber product, separator, secondary battery, electric double layer capacitor, and method for producing nonwoven fabric 东丽株式会社 2022-04-29 CN disclosed
EP-3650481-A1 RESIN, RESIN COMPOSITION, NONWOVEN FABRIC USING SAME, FIBER PRODUCT, SEPARATOR, SECONDARY BATTERY, AND METHOD FOR PRODUCING ELECTRIC DOUBLE LAYER CAPACITOR AND NONWOVEN FABRIC Toray Industries, Inc. (JP) 2020-05-13 EP disclosed
US-20200131366-A1 RESIN, RESIN COMPOSITION, NONWOVEN FABRIC USING SAME, FIBER PRODUCT, SEPARATOR, SECONDARY BATTERY AND ELECTRIC DOUBLE LAYER CAPACITOR, AND METHOD FOR PRODUCING NONWOVEN FABRIC TORAY INDUSTRIES, INC. (JP) 2020-04-30 US disclosed
CN-110799559-A Resin, resin composition, nonwoven fabric, fiber product, separator, secondary battery, electric double layer capacitor, and method for producing nonwoven fabric 东丽株式会社 2020-02-14 CN disclosed