SCHEMBL2219655

SCHEMBL2219655

Cc1cccc([N+](=O)[O-])c1[N+](=O)[O-].O=[N+]([O-])[O-].[Na+]

nearest known ligand 0.92

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.92
TDP1 Q9NUW8 5/20 0.69
ALDH1A1 P00352 4/20 0.69
SMN1; SMN2 Q16637 1/20 0.62
HSD17B10 Q99714 1/20 0.61
GPR35 Q9HC97 2/20 0.55
L3MBTL1 Q9Y468 2/20 0.53
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.44
KAT2B Q92831 1/20 0.43
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 1/20 0.42
S100A4 P26447 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1101208 0.96 TSHR (1.00) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL146895 0.96 TSHR (1.00) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL29359563 0.96 TSHR (1.00) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL11696134 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
Magnesium SCHEMBL11696142 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL8717819 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL28589645 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL31188803 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
Fluoride SCHEMBL28054250 0.94 TSHR (0.96) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10
O-Xylene SCHEMBL28588420 0.92 TSHR (0.92) TSHRTDP1ALDH1A1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1854160-A2 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2007-11-14 EP claimed
WO-2006085319-A2 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT COMPANY LTD. (IL) 2006-08-17 WO claimed
EP-3228624-A2 REDOX-ACTIVE CHROMOPHORE MOLECULES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2017-10-11 EP disclosed
US-9309274-B2 Redox-active structures and devices utilizing the same YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2016-04-12 US disclosed
US-20150007371-A1 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2015-01-01 US disclosed
US-8865890-B2 Redox-active structures and devices utilizing the same YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2014-10-21 US disclosed
US-20140196180-A1 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH & DEVELOPMENT COMPANY LTD. (IL) 2014-07-10 US disclosed
US-8722879-B2 Redox-active structures and devices utilizing the same YEDA RESEARCH & DEVELOPMENT COMPANY LTD. AT THE WEIZMANN INSTITUTE OF SCIENCE (IL) 2014-05-13 US disclosed
US-20110177964-A1 CHEMOSENSORY ARRAYS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2011-07-21 US disclosed
EP-1854160-A2 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2007-11-14 EP disclosed
US-20070258147-A1 Redox-active structures and devices utilizing the same YEDA RESEARCH & DEVELOPMENT CO., LTD. (IL) 2007-11-08 US disclosed
WO-2006085319-A2 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME YEDA RESEARCH AND DEVELOPMENT COMPANY LTD. (IL) 2006-08-17 WO disclosed
US-6610977-B2 Security system for NBC-safe building LOCKHEED MARTIN CORPORATION 2003-08-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140196180-A1 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME GPX4, GPX1, LPO TSHR 4361/4885TDP1 2760/4885ALDH1A1 233/4885
US-20150007371-A1 REDOX-ACTIVE STRUCTURES AND DEVICES UTILIZING THE SAME GPX4, GPX1, LPO TSHR 4361/4885TDP1 2760/4885ALDH1A1 233/4885
US-20070258147-A1 Redox-active structures and devices utilizing the same GPX4, GPX1, LPO TSHR 4361/4885TDP1 2760/4885ALDH1A1 233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.