Tiron

Tiron

SCHEMBL22220

O=S(=O)([O-])c1cc(O)c(O)c(S(=O)(=O)[O-])c1.[Na+].[Na+]

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Tiron. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 1/20 0.42
CA12 known ✓ O43570 1/20 0.38
CA1 known ✓ P00915 1/20 0.38
CA2 known ✓ P00918 1/20 0.38
THRB known ✓ P10828 1/20 0.36
DUSP5 Q16690 4/20 0.65
PTPN1 P18031 5/20 0.57
DUSP6 Q16828 1/20 0.52
PKLR P30613 5/20 0.45
SIRT1 Q96EB6 1/20 0.41
PRMT1 Q99873 1/20 0.41
APP P05067 1/20 0.41
PGAM1 P18669 2/20 0.41
POLB P06746 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
GRK2 P25098 1/20 0.40
PLEC Q15149 1/20 0.40
PLCG1 P19174 1/20 0.39
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tiron SCHEMBL29385574 1.00 DUSP5 (0.65) DUSP5PTPN1DUSP6PKLRPTGS1
SCHEMBL5310574 1.00 DUSP5 (0.65) DUSP5PTPN1DUSP6PKLRPTGS1
Water SCHEMBL5097417 0.98 DUSP5 (0.62) DUSP5PTPN1DUSP6PKLRPTGS1
Water SCHEMBL29379961 0.98 DUSP5 (0.62) DUSP5PTPN1DUSP6PKLRPTGS1
Water SCHEMBL3205313 0.98 DUSP5 (0.62) DUSP5PTPN1DUSP6PKLRPTGS1
SCHEMBL10722008 0.98 DUSP5 (0.62) DUSP5PTPN1DUSP6PKLRPTGS1
Ammonia Solution, Strong SCHEMBL9751555 0.98 DUSP5 (0.62) DUSP5PTPN1DUSP6PKLRPTGS1
SCHEMBL31393 0.96 DUSP5 (0.59) DUSP5PTPN1DUSP6PKLRPTGS1
Potassium Ion SCHEMBL3222667 0.96 DUSP5 (0.59) DUSP5PTPN1DUSP6PKLRPTGS1
SCHEMBL9328871 0.96 DUSP5 (0.59) DUSP5PTPN1DUSP6PKLRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6575 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090621-A1 SYSTEMS, DEVICES, AND METHODS FOR SEPARATION OF METALS FROM WASTE, SCRAP, AND POST-CONSUMER PRODUCTS SUNCHEM INC. (US) 2026-04-30 WO claimed
EP-3301162-B1 LOW PH LAUNDRY DETERGENT COMPOSITION PROCTER & GAMBLE (US) 2026-04-15 EP claimed
EP-3301163-B1 LOW PH LAUNDRY DETERGENT COMPOSITION PROCTER & GAMBLE (US) 2026-04-15 EP claimed
EP-3301164-B1 LOW PH LAUNDRY DETERGENT COMPOSITION PROCTER & GAMBLE (US) 2026-04-15 EP claimed
EP-4206645-B1 METHOD AND APPARATUS FOR REMOVING OR REDUCING FORMATION OF PRECIPITATES GENERATED IN HEMATOXYLIN SOLUTIONS VENTANA MED SYST INC (US) 2026-03-11 EP claimed
EP-4699720-A2 FOUNDRY SLIP Safran (FR) 2026-02-25 EP claimed
EP-3684525-B1 USE OF A CASTING SLURRY SAFRAN (FR) 2026-02-18 EP claimed
US-12533430-B2 Metal nuclide-loaded carbon microsphere (CMS), preparation method, and use thereof Chengdu New Radiomedicine Technology Co., Ltd. (CN) 2026-01-27 US claimed
EP-4665689-A1 ANTISCALANT COMPOSITIONS AND METHODS OF USE Locus Solutions IPCO, LLC (US) 2025-12-24 EP claimed
EP-3301151-B1 LOW PH LAUNDRY DETERGENT COMPOSITION PROCTER & GAMBLE (US) 2025-11-12 EP claimed
US-5302531-A Mixture of complexing agent, metal compound and indicator MILES INC. (US) 1994-04-12 US claimed
WO-1994001142-A1 THERAPEUTIC COMPOSITIONS AND METHODS USING PQQ THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 1994-01-20 WO claimed
US-5242832-A Surfactants and hemoglobin stabilizers TOA MEDICAL ELECTRONICS CO., LTD. (JP) 1993-09-07 US claimed
WO-1993014751-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING AS ACTIVE PRINCIPLE ASSOCIATIONS OF VANADIUM AND/OR NIOBIUM WITH PYROCATECHOL DERIVATIVES I.R.2.M. (FR) 1993-08-05 WO claimed
EP-0444241-A1 Reagent for measurement of leukocytes and hemoglobin in blood TOA MEDICAL ELECTRONICS CO., LTD. (JP) 1991-09-04 EP claimed
US-4714614-A PSEUDOMONAS AND FERRIC ION CHELATING AGENT COLORADO STATE UNIVERSITY (US) 1987-12-22 US claimed
US-4279870-A Liquid-liquid extraction process for the recovery of tungsten from low level sources GTE LABORATORIES INCORPORATED (US) 1981-07-21 US claimed
US-4264716-A STABILIZED BY ADDITION OF AN AMINOPOLYPHOSPHONIC ACID SEQUESTERING AGENT EASTMAN KODAK COMPANY (US) 1981-04-28 US claimed
US-4194954-A Electrolytic etch preparation of semiconductor surfaces THE POST OFFICE (GB) 1980-03-25 US claimed
US-4112044-A CATALYTIC ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1978-09-05 US claimed