SCHEMBL2273998

SCHEMBL2273998

O=C(O)c1ccc(-c2ccccc2)cc1NC(=O)c1cn[nH]c1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACLY P53396 11/20 0.55
TDP1 Q9NUW8 1/20 0.49
DHODH Q02127 1/20 0.47
DCAF1 Q9Y4B6 1/20 0.46
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
MEN1 O00255 1/20 0.44
GFER P55789 1/20 0.44
KMT2A Q03164 1/20 0.44
SUCNR1 Q9BXA5 1/20 0.44
HDAC1 Q13547 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
GRIK1 P39086 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2270261 0.85 CYP2C9 (0.46) TDP1DCAF1MEN1GFERKMT2A
SCHEMBL1672584 0.81 TDP1 (0.63) ACLYTDP1DHODHDCAF1KDM5B
SCHEMBL27696872 0.78 HSP90AA1 (0.62) TDP1DCAF1HSP90AA1HSP90AB1MEN1
SCHEMBL28059476 0.78 LMNA (0.51) DCAF1KDM5B
SCHEMBL2268189 0.78 ACLY (0.61) ACLYDHODHSUCNR1HDAC1
SCHEMBL1320352 0.77 ACMSD (0.68) ACLYDHODHMEN1GFERKMT2A
SCHEMBL2270222 0.77 DHODH (0.77) ACLYTDP1DHODHMEN1KMT2A
SCHEMBL2275453 0.77 ACLY (0.76) ACLYTDP1DHODHMEN1KMT2A
SCHEMBL1317052 0.76 ACLY (0.64) ACLYDHODHMEN1KMT2ASUCNR1
SCHEMBL2275016 0.76 TP53 (0.58) ACLYTDP1DHODHHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 ACLY 653/4885TDP1 3823/4885DHODH 1469/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.