SCHEMBL2566447

SCHEMBL2566447

CC(=O)c1ccc(F)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.46
KCNQ3 O43525 1/20 0.44
KCNQ2 O43526 1/20 0.44
EPHX2 P34913 1/20 0.43
HPGD P15428 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
MAOB P27338 1/20 0.40
BDKRB1 P46663 1/20 0.39
P4HA1 P13674 1/20 0.39
P4HTM Q9NXG6 1/20 0.39
HSD17B1 P14061 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2B6 P20813 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15274452 1.00 KCNJ1 (0.46) KCNJ1KCNQ3KCNQ2EPHX2HPGD
SCHEMBL29790306 1.00 KCNJ1 (0.46) KCNJ1KCNQ3KCNQ2EPHX2HPGD
SCHEMBL483725 0.84 HSD17B1 (0.52) MAPTLMNAMAOBHSD17B1SMN1; SMN2
SCHEMBL27594193 0.82 RXFP1 (0.53) KCNQ3KCNQ2EPHX2HPGDMAPT
Acetic Acid SCHEMBL28599450 0.80 NNMT (0.53) EPHX2L3MBTL1SMN1; SMN2
SCHEMBL646556 0.80 P4HA1 (0.61) EPHX2HPGDL3MBTL1MAPTP4HA1
SCHEMBL29723813 0.80 P4HA1 (0.61) EPHX2HPGDL3MBTL1MAPTP4HA1
SCHEMBL29646483 0.80 P4HA1 (0.61) EPHX2HPGDL3MBTL1MAPTP4HA1
SCHEMBL30448953 0.80 P4HA1 (0.61) EPHX2HPGDL3MBTL1MAPTP4HA1
SCHEMBL18910409 0.78 KCNQ3 (0.44) KCNQ3KCNQ2EPHX2HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 99 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244728-B1 USE OF HETEROARYLETHYL AMINES TO STIMULATE ANIMAL GROWTH, HETEROARYLETHYL AMINES AND PROCESS FOR THEIR PREPARATION BAYER AG (DE) 1992-11-11 EP claimed
US-20260041671-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS INC (US) 2026-02-12 US disclosed
US-12539292-B2 BRM targeting compounds and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-02-03 US disclosed
EP-4537905-A2 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE Arvinas Operations, Inc. (US) 2025-04-16 EP disclosed
EP-3774789-B1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS INC (US) 2025-03-05 EP disclosed
US-20250042911-A1 NOVEL BENZOPYRAN DERIVATIVE AND USE THEREOF SPARK BIOPHARMA, INC. (KR) 2025-02-06 US disclosed
CN-113135896-B Methylpyrazole derivatives as RET inhibitors 正大天晴药业集团股份有限公司 2024-12-06 CN disclosed
US-20240327417-A1 HETEROCYCLIC COMPOUNDS BEIGENE SWITZERLAND GMBH (CH) 2024-10-03 US disclosed
CN-112654621-B Substituted naphthyridinone compounds useful as T cell activators 百时美施贵宝公司 2024-05-14 CN disclosed
EP-4365175-A1 NOVEL BENZOPYRAN DERIVATIVE AND USE THEREOF Spark Biopharma, Inc. (KR) 2024-05-08 EP disclosed
US-5001138-A Insecticides NIHON TOKUSHU NOYAKU SEIZO, K.K. (JP) 1991-03-19 US disclosed
US-4845106-A INSECTICIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-07-04 US disclosed
US-4816457-A HYPOTENSIVE AGENTS, BRONCHODILATORS, EYES MERCK & CO., INC., A CORP. OF NJ 1989-03-28 US disclosed
US-4742060-A 2-(NITROIMINO)- OR 2-(NITROMETHYLENE)-IMIDAZOLIDINES AS INSECTICIDES NIHON TOKUSHU NOYAKU SEIZO K. K. (JP) 1988-05-03 US disclosed
EP-0105053-B1 ARALKYLAMINOETHANOL HETEROCYCLIC COMPOUNDS MERCK & CO. INC. (US) 1988-01-20 EP disclosed
EP-0244728-A2 Use of heteroarylethyl amines to stimulate animal growth, heteroarylethyl amines and process for their preparation BAYER AG (DE) 1987-11-11 EP disclosed
US-4686222-A ADRENERGIC BLOCKERS, BRONCHODILATORS MERCK & CO., INC. (US) 1987-08-11 US disclosed
EP-0192060-A1 Heterocyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1986-08-27 EP disclosed
US-4568679-A ADRENERGIC BLOCKING AGENTS, HYPOTENSIVE AGENTS, BRONCHODILATOR AGENTS, REDUCING INTRAOCULAR PRESSURE MERCK & CO., INC. (US) 1986-02-04 US disclosed
EP-0105053-A1 Aralkylaminoethanol heterocyclic compounds MERCK & CO. INC. (US) 1984-04-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12539292-B2 BRM targeting compounds and associated methods of use ADRM1, SUMO2, BAZ1A KCNJ1 4799/4885KCNQ3 4750/4885KCNQ2 4770/4885
US-20240327417-A1 HETEROCYCLIC COMPOUNDS NFATC1, CD4, ACIN1 KCNJ1 3989/4885KCNQ3 4810/4885KCNQ2 4649/4885
US-20250042911-A1 NOVEL BENZOPYRAN DERIVATIVE AND USE THEREOF MYD88, MYADM, CD14 KCNJ1 3261/4885KCNQ3 4692/4885KCNQ2 4725/4885
US-20260041671-A1 BRM TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ADRM1, VHL, BAZ1A KCNJ1 4685/4885KCNQ3 4573/4885KCNQ2 4682/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.