SCHEMBL257249

SCHEMBL257249

CCc1cc(Br)ccc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
GLA P06280 1/20 0.50
POLB P06746 1/20 0.46
MYC P01106 1/20 0.46
NR4A1 P22736 1/20 0.46
RXFP1 Q9HBX9 3/20 0.45
PRNP P04156 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PPARG P37231 1/20 0.45
HIF1A Q16665 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NR2E3 Q9Y5X4 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
GABRP O00591 2/20 0.44
GABRD O14764 2/20 0.44
GABRA1 P14867 2/20 0.44
GABRB1 P18505 2/20 0.44
GABRG2 P18507 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3206015 0.87 POLB (0.47) KDM4EGLAPOLBMYCNR4A1
SCHEMBL696316 0.85 ALDH1A1 (0.50) KDM4EGLAPOLBMYCNR4A1
SCHEMBL3746157 0.84 PTGDR2 (0.53) KDM4EGLAPOLBMYCNR4A1
SCHEMBL31125276 0.84 KDM4E (0.55) KDM4EGLAPOLBMYCNR4A1
SCHEMBL1500169 0.84 KDM4E (0.50) KDM4EGLAPOLBMYCNR4A1
SCHEMBL23243427 0.84 KDM4E (0.55) KDM4EGLAPOLBMYCNR4A1
SCHEMBL6513432 0.84 HSD17B1 (0.56) RXFP1PRNPCYP1A2CYP2C9CYP2C19
SCHEMBL11151739 0.84 GABRP (0.51) KDM4EGLAPOLBMYCNR4A1
SCHEMBL29907952 0.83 NHERF1 (0.49) KDM4EPOLBCYP1A2CYP2C9CYP2C19
SCHEMBL1674351 0.83 KDM4E (0.46) KDM4EGLAPOLBMYCNR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 525 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116891448-A Preparation method of roflumilast intermediate III 上海医药集团青岛国风药业股份有限公司 2023-10-17 CN claimed
EP-2516479-B1 NEW INTERNAL AND EXTERNAL DONOR COMPOUNDS FOR OLEFIN POLYMERIZATION CATALYSTS BASF CORP (US) 2016-04-20 EP claimed
US-8569195-B2 Internal and external donor compounds for olefin polymerization catalysts II BASF CORPORATION (US) 2013-10-29 US claimed
EP-2516479-A2 NEW INTERNAL AND EXTERNAL DONOR COMPOUNDS FOR OLEFIN POLYMERIZATION CATALYSTS BASF Corporation (US) 2012-10-31 EP claimed
US-8211819-B2 Internal and external donor compounds for olefin polymerization catalysts BASF CORPORATION (US) 2012-07-03 US claimed
WO-2011084691-A2 NEW INTERNAL AND EXTERNAL DONOR COMPOUNDS FOR OLEFIN POLYMERIZATION CATALYSTS BASF CORPORATION (US) 2011-07-14 WO claimed
US-20110152481-A1 Internal and external donor compounds for olefin polymerization catalysts BASF CATALYSTS LLC (US) 2011-06-23 US claimed
US-20260078130-A1 NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF SIRONAX LTD (KY) 2026-03-19 US disclosed
US-12551490-B2 Heterocyclic modulators of lipid synthesis SAGIMET BIOSCIENCES INC. (US) 2026-02-17 US disclosed
CN-116891448-B Preparation method of roflumilast intermediate III 上海医药集团青岛国风药业股份有限公司 2026-02-03 CN disclosed
US-20260015743-A1 MEDIATED HYDROGEN ANODE FOR USE IN REDUCTIVE ELECTROSYNTHESIS WISCONSIN ALUMNI RES FOUND (US) 2026-01-15 US disclosed
US-20250368620-A1 ARNT Degrading Compounds and Uses Thereof CELGENE CORPORATION (US) 2025-12-04 US disclosed
US-12448368-B2 Indole compounds as androgen receptor modulators NIDO BIOSCIENCES, INC. (US) 2025-10-21 US disclosed
EP-0206635-A1 Preparation of 3-amino-4-hydroxybenzoic acids THE DOW CHEMICAL COMPANY (US) 1986-12-30 EP disclosed
US-4526882-A Contacting magnesium alcoholate and group II or group IIIA metal alkyl, treating with titanium halide and electron donor, comminuting, treating product with titanium halide, ethyl benzoate, aromatic acid ester STANDARD OIL COMPANY (INDIANA) (US) 1985-07-02 US disclosed
US-4316853-A Insecticidal tetraorganotin compounds M&T CHEMICALS INC. (US) 1982-02-23 US disclosed
EP-0001717-B1 INSECTICIDAL COMPOSITIONS CONTAINING TETRAORGANOTIN COMPOUNDS AND METHOD FOR USING SAME M & T CHEMICALS, INC. (US) 1981-11-04 EP disclosed
US-4212810-A INSECTICIDES M&T CHEMICALS INC. (US) 1980-07-15 US disclosed
EP-0001717-A2 Insecticidal compositions containing tetraorganotin compounds and method for using same M & T CHEMICALS, INC. (US) 1979-05-02 EP disclosed
US-4138483-A Insecticidal compositions containing certain tetraorganotin compounds and method for using same M&T CHEMICALS INC. (US) 1979-02-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260015743-A1 MEDIATED HYDROGEN ANODE FOR USE IN REDUCTIVE ELECTROSYNTHESIS HAO2, HACL2, HVCN1 KDM4E 3823/4885GLA 3260/4885POLB 1207/4885
US-20260078130-A1 NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF NAMPT, NNMT, SARM1 KDM4E 3382/4885GLA 2057/4885POLB 1690/4885
US-12551490-B2 Heterocyclic modulators of lipid synthesis FASN, FADS1, FADS2 KDM4E 1054/4885GLA 4205/4885POLB 3427/4885
US-12448368-B2 Indole compounds as androgen receptor modulators AR, FSHR, ADRB3 KDM4E 1533/4885GLA 2251/4885POLB 2183/4885
US-20250368620-A1 ARNT Degrading Compounds and Uses Thereof ARNT, AHR, NR1H2 KDM4E 2453/4885GLA 2084/4885POLB 2188/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.