SCHEMBL2598448

SCHEMBL2598448

CCn1ncc2nccc(I)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.40
HASPIN Q8TF76 1/20 0.36
PDE1A P54750 3/20 0.34
PDE1B Q01064 3/20 0.34
PDE1C Q14123 3/20 0.34
HTT P42858 1/20 0.33
CLK1 P49759 1/20 0.32
DYRK1A Q13627 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
APOBEC3A P31941 1/20 0.31
BLM P54132 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CCNK O75909 1/20 0.31
CDK12 Q9NYV4 1/20 0.31
CYP11B2 P19099 1/20 0.30
XDH P47989 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2598467 0.87 ADORA3 (0.38) TGFBR1PDE1APDE1BPDE1CPOLB
SCHEMBL2598377 0.80 MPO (0.35) TGFBR1KDM4EALDH1A1
SCHEMBL2598326 0.79 TTBK1 (0.33) TGFBR1
SCHEMBL2598465 0.78 TGFBR1 (0.39) TGFBR1KDM4EALDH1A1
SCHEMBL2598357 0.77 MAPK1 (0.33) TGFBR1DYRK1AALDH1A1
SCHEMBL2598332 0.77 TGFBR1 (0.37) TGFBR1ALDH1A1POLB
SCHEMBL2598351 0.75 NPBWR1 (0.49) KDM4EALDH1A1
SCHEMBL2598302 0.75 DGAT1 (0.32)
SCHEMBL2598306 0.72 PDE1B (0.34) PDE1APDE1BPDE1CCLK1DYRK1A
SCHEMBL2598490 0.71 ALDH1A1 (0.36) KDM4EALDH1A1GAABLMCCNK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146287-A1 PYRAZOLO[4,3-B]PYRIDINE-7-AMINE INHIBITORS OF ALK5 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-11-24 WO disclosed