SCHEMBL27248243

SCHEMBL27248243

O=C1CCON1Cc1cccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
KCNN4 O15554 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
CA2 P00918 1/20 0.41
FAAH O00519 1/20 0.40
CYP11B1 P15538 1/20 0.40
ADRA2C P18825 1/20 0.40
CYP11B2 P19099 1/20 0.40
MBTD1 Q05BQ5 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
MAOB P27338 1/20 0.39
XDH P47989 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847449 0.80 L3MBTL1 (0.45) SMN1; SMN2KDM4EMEN1KMT2A
SCHEMBL44669 0.80 L3MBTL1 (0.45) SMN1; SMN2KDM4EMEN1KMT2A
SCHEMBL5766288 0.76 SMN1; SMN2 (0.53) SMN1; SMN2TDP1CA12CA9KCNN4
SCHEMBL9762141 0.71 KDM4E (0.39) CA9CYP11B1CYP11B2KDM4EMEN1
SCHEMBL18763113 0.71 ALDH1A1 (0.44) MEN1KMT2A
SCHEMBL3388088 0.71 L3MBTL1 (0.58) SMN1; SMN2TDP1KCNN4FAAHMBTD1
SCHEMBL3994597 0.71 SMN1; SMN2 (0.48) SMN1; SMN2TDP1CA12CA9KCNN4
SCHEMBL29067018 0.70 SMN1; SMN2 (0.68) SMN1; SMN2TDP1FAAHMBTD1L3MBTL3
SCHEMBL22815820 0.70 L3MBTL1 (0.65) SMN1; SMN2TDP1FAAHMBTD1L3MBTL3
SCHEMBL9760860 0.69 LOXL2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12404253-B2 2,4,6-trisubstituted 1,3,5-triazines as modulators of CX3CR1 ASTRAZENECA AB (SE) 2025-09-02 US disclosed
EP-4605388-A1 <SUP2/>? <SUB2/>?3?2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CXCR1 Astrazeneca AB (SE) 2025-08-27 EP disclosed
US-20240383866-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 ASTRAZENECA AB (SE) 2024-11-21 US disclosed
US-20240199558-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 ASTRAZENECA AB (SE) 2024-06-20 US disclosed
WO-2024083933-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX 3CR1 ASTRAZENECA AB (SE) 2024-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240199558-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 CX3CR1, CCR2, CCR5 SMN1; SMN2 1048/4885TDP1 2513/4885CA12 4722/4885
US-20240383866-A1 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES AS MODULATORS OF CX3CR1 CX3CR1, CCR2, CCR5 SMN1; SMN2 1048/4885TDP1 2513/4885CA12 4722/4885
US-12404253-B2 2,4,6-trisubstituted 1,3,5-triazines as modulators of CX3CR1 CX3CR1, CCR2, CCR5 SMN1; SMN2 1048/4885TDP1 2513/4885CA12 4722/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.