SCHEMBL28025013

SCHEMBL28025013

CCN(CC)c1ccc(N=Nc2ccc(Br)cn2)c(O)c1.[Na+].c1ccc([B-](c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.44

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.44
RIOK2 Q9BVS4 1/20 0.40
MAPT P10636 5/20 0.37
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 2/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 1/20 0.36
NPC1 O15118 2/20 0.35
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL272969 0.89 KCNH2 (0.47) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL272970 0.89 KCNH2 (0.47) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL29397508 0.89 KCNH2 (0.47) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL29397420 0.89 KCNH2 (0.47) KCNH2RIOK2MAPTKDM4EALDH1A1
Bromide SCHEMBL30705401 0.88 KCNH2 (0.48) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL8206882 0.88 KCNH2 (0.46) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL14484276 0.78 KCNH2 (0.43) KCNH2RIOK2MAPTKDM4EALDH1A1
SCHEMBL4343598 0.77 KCNH2 (0.64) KCNH2RIOK2MAPTALDH1A1SMN1; SMN2
SCHEMBL4343601 0.77 KCNH2 (0.64) KCNH2RIOK2MAPTALDH1A1SMN1; SMN2
SCHEMBL8654656 0.76 KCNH2 (0.47) KCNH2RIOK2MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105136694-A Method for determining trace copper, trace zinc and trace iron in mineral water through ion pair-cloud point extraction- cloud point extraction-flame atomic absorption spectrometry UNIV GUANGDONG PHARM 2015-12-09 CN claimed
CN-105136694-A Method for determining trace copper, trace zinc and trace iron in mineral water through ion pair-cloud point extraction- cloud point extraction-flame atomic absorption spectrometry UNIV GUANGDONG PHARM 2015-12-09 CN disclosed