SCHEMBL28073660

SCHEMBL28073660

C=Cc1ccc2c(CCOC(C)=O)csc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.37
ITGB1 P05556 1/20 0.37
ITGAV P06756 1/20 0.37
ITGA5 P08648 1/20 0.37
ITGB5 P18084 1/20 0.37
MTNR1A P48039 11/20 0.36
MTNR1B P49286 6/20 0.36
TKT P29401 1/20 0.32
LMNA P02545 1/20 0.32
RAD52 P43351 1/20 0.32
HTR2C P28335 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27752659 0.82 ITGB3 (0.39) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL28073641 0.80 PKM (0.39) LMNAALDH1A1PPARGPPARDPPARA
SCHEMBL28693243 0.77 CYP2A6 (0.53) MTNR1ARAD52ALDH1A1
SCHEMBL28073664 0.71 LRRK2 (0.33) ALDH1A1
SCHEMBL8592477 0.70 MET (0.46) LMNAALDH1A1
SCHEMBL8132867 0.70 MTNR1A (0.67) MTNR1AMTNR1BHTR2C
Water SCHEMBL27600001 0.69 MET (0.45) LMNAALDH1A1
SCHEMBL28073642 0.69 ALOX15 (0.40) LMNAALDH1A1
SCHEMBL16693174 0.67 CYP2A6 (0.42) LMNAALDH1A1
SCHEMBL5549982 0.66 CHRNB2 (0.51) LMNAALDH1A1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254525-B aromatic ring compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-05-25 CN disclosed