Cloprostenol

Cloprostenol

SCHEMBL28077016

O=C([O-])CCC/C=C\C[C@@H]1C(/C=C/[C@@H](O)COc2cccc(Cl)c2)[C@H](O)C[C@@H]1O.[Na+]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cloprostenol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
THRB known ✓ P10828 1/20 0.84
ABCC4 O15439 2/20 1.00
PTGFR P43088 16/20 0.84
PTGER3 P43115 5/20 0.84
TBXA2R P21731 2/20 0.84
PTGER1 P34995 2/20 0.84
PTGER2 P43116 1/20 0.84
ABCB11 O95342 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cloprostenol SCHEMBL29600088 1.00 ABCC4 (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL28242 1.00 ABCC4 (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL29709332 1.00 ABCC4 (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL28850753 1.00 ABCC4 (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Delprostenate SCHEMBL8206607 0.92 ABCC4 (0.84) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL17200671 0.92 PTGFR (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL15390430 0.92 PTGFR (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL123595 0.92 PTGFR (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL123596 0.92 PTGFR (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1
Cloprostenol SCHEMBL14913508 0.92 PTGFR (1.00) ABCC4PTGFRPTGER3TBXA2RPTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117941651-A Method for improving lambing rate and/or gestation rate of sheep and composition used by method 中国农业大学 2024-04-30 CN disclosed
CN-105755944-A Bridge construction method 张译元 2016-07-13 CN disclosed
CN-105714687-A Building method for bridge 武汉理工大学 2016-06-29 CN disclosed