SCHEMBL2855477

SCHEMBL2855477

C=C(C)c1ccccc1NC(=O)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GPR6 P46095 1/20 0.38
TRPC1 P48995 1/20 0.37
TRPC3 Q13507 1/20 0.37
STIM1 Q13586 1/20 0.37
ORAI1 Q96D31 1/20 0.37
STIM2 Q9P246 1/20 0.37
ACHE P22303 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CCR1 P32246 4/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
NR3C1 P04150 1/20 0.35
P2RY1 P47900 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853031 0.89 MAPT (0.41) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2859508 0.86 CYP1A2 (0.46) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2852552 0.86 MEN1 (0.51) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2848541 0.85 RAB9A (0.43) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2854596 0.85 TP53 (0.46) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850855 0.85 KEAP1 (0.36) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850388 0.85 LMNA (0.35) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2850610 0.85 MAPT (0.40) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2857074 0.84 LPAR1 (0.42) MAPTPOLBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2855775 0.83 P2RY1 (0.44) MAPTPOLBSMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed