SCHEMBL2857337

SCHEMBL2857337

O=C(Nc1cccc(F)c1)Oc1cnn(-c2ncccn2)c1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 3/20 0.43
HSP90AA1 P07900 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
P2RY1 P47900 1/20 0.41
MTOR P42345 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
CD38 P28907 2/20 0.39
CDK8 P49336 1/20 0.39
MALT1 Q9UDY8 1/20 0.38
LRRK2 Q5S007 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854810 0.89 KMT2A (0.46) KMT2AMEN1MAPTHSP90AA1KDM4E
SCHEMBL2855496 0.87 KDM4E (0.46) KMT2AMEN1MAPTHSP90AA1KDM4E
SCHEMBL2854269 0.86 RAB9A (0.46) MAPTNPC1RAB9ALMNAMTOR
SCHEMBL2854592 0.85 MEN1 (0.40) KMT2AMEN1MAPTHSP90AA1KDM4E
SCHEMBL2854572 0.84 RAB9A (0.44) KMT2AMEN1MAPTHSP90AA1KDM4E
SCHEMBL2854492 0.83 MAPT (0.42) KMT2AMEN1MAPTHSP90AA1KDM4E
SCHEMBL2861646 0.82 NPC1 (0.42) KMT2AMEN1MAPTKDM4ENPSR1
SCHEMBL2861607 0.81 TRPV1 (0.42) KMT2AMEN1L3MBTL1P2RY1
SCHEMBL2855950 0.80 POLB (0.41) MAPTKDM4ENPC1RAB9ALMNA
SCHEMBL2850733 0.78 KEAP1 (0.46) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed