SCHEMBL2860103

SCHEMBL2860103

CCN(CC)C(=O)c1cccc(NC(=O)Oc2cnn(-c3ccccc3)c2C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.44
KEAP1 Q14145 2/20 0.43
NFE2L2 Q16236 2/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
BRAF P15056 1/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
CYP1A2 P05177 1/20 0.40
PDE11A Q9HCR9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860210 0.92 NR3C1 (0.42) NR3C1KEAP1NFE2L2RAB9ASMN1; SMN2
SCHEMBL2857883 0.85 MAPT (0.44) RAB9ANPC1SMN1; SMN2ALDH1A1POLB
SCHEMBL2850725 0.82 MAPT (0.54) KEAP1NFE2L2NPC1SMN1; SMN2KDM4E
SCHEMBL2854287 0.82 MAPT (0.52) NR3C1KEAP1NFE2L2RAB9ASMN1; SMN2
SCHEMBL2862974 0.80 KEAP1 (0.50) KEAP1NFE2L2RAB9ANPC1SMN1; SMN2
SCHEMBL2860939 0.80 LMNA (0.45) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL2857954 0.79 RAB9A (0.53) NR3C1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL2848492 0.79 ALDH1A1 (0.47) KEAP1NFE2L2SMN1; SMN2KDM4EALDH1A1
SCHEMBL2858122 0.78 MAPT (0.53) SMN1; SMN2KDM4EALDH1A1POLBMAPT
SCHEMBL2860829 0.77 TNKS (0.42) SMN1; SMN2KDM4EALDH1A1BRAFMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed