SCHEMBL28844707

SCHEMBL28844707

COc1cc(Nc2cc(Cl)cc3[nH]cc(C(C)OC=O)c23)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.38
TDO2 P48775 5/20 0.38
P2RY4 P51582 1/20 0.36
GRM4 Q14833 3/20 0.34
KCNH2 Q12809 1/20 0.32
TGFBR1 P36897 1/20 0.31
P2RX7 Q99572 2/20 0.31
EGFR P00533 1/20 0.31
BUB1 O43683 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28338822 0.78 IDO1 (0.34) IDO1TDO2
SCHEMBL28338774 0.76 PTGS2 (0.35) IDO1TDO2EGFRMTNR1AMTNR1B
SCHEMBL28880740 0.74 PTGS2 (0.43) IDO1TDO2EGFR
SCHEMBL27309524 0.73 GPR17 (0.39) MTNR1AMTNR1B
SCHEMBL28168774 0.71 PTK6 (0.41) GRM4EGFRMTNR1AMTNR1B
SCHEMBL27694363 0.71 GPR84 (0.32)
SCHEMBL29865098 0.70 P2RX7 (0.51) IDO1TDO2P2RY4GRM4KCNH2
Ethoxycarbonyl Group SCHEMBL28844709 0.70 P2RX7 (0.47) IDO1TDO2P2RY4GRM4P2RX7
SCHEMBL27908784 0.68 MTNR1A (0.43) EGFRMTNR1AMTNR1B
SCHEMBL28291585 0.68 ALDH1A1 (0.37) EGFRMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed