SCHEMBL29005254

SCHEMBL29005254

CON(C)C(=O)c1ccc(OC(F)C(F)F)nn1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.40
MLYCD O95822 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29005279 0.78 SIRT6 (0.39) MLYCD
SCHEMBL29005296 0.77 NNMT (0.40) NNMT
SCHEMBL29005252 0.74 L3MBTL1 (0.43) NNMTMLYCD
SCHEMBL30342225 0.74 L3MBTL1 (0.43) NNMTMLYCD
SCHEMBL24724207 0.72 MLYCD (0.37) NNMTMLYCDTRPM8
SCHEMBL30003812 0.72 MLYCD (0.37) NNMTMLYCDTRPM8
SCHEMBL2541582 0.71 PKM (0.39) NNMTMLYCDTRPM8
SCHEMBL15142310 0.69 NNMT (0.61) NNMT
SCHEMBL29162132 0.68 TRPM8 (0.38) MLYCDTRPM8
SCHEMBL29106396 0.67 MEN1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134018-A 2-oxoimidazolidine-4-carboxamide as NAV1.8 inhibitor 默沙东有限责任公司 2023-05-16 CN disclosed
CN-116056697-A 2-oxo-oxazolidine-5-carboxamides as NAV1.8 inhibitors 默沙东有限责任公司 2023-05-02 CN disclosed