SCHEMBL29028690

SCHEMBL29028690

N#CCc1c2ccc(F)cc2nn1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.39
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
CSNK1A1 P48729 1/20 0.36
CDK8 P49336 1/20 0.36
NEK2 P51955 1/20 0.36
LIMK1 P53667 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
KDM4E B2RXH2 3/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PDE10A Q9Y233 2/20 0.36
GRM4 Q14833 1/20 0.35
MAPK1 P28482 3/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
HSD17B10 Q99714 2/20 0.35
ALOX15 P16050 1/20 0.35
MCL1 Q07820 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29028699 0.84 MEN1 (0.39) MAPTCHEK1AURKACSNK1A1CDK8
SCHEMBL29028696 0.84 CSNK2A1 (0.40) MAPTCHEK1AURKACSNK1A1CDK8
SCHEMBL29028719 0.83 MAPT (0.46) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL29028700 0.83 MPO (0.47) MAPTKDM4EMAPK1ALDH1A1HPGD
SCHEMBL29028720 0.83 ADORA3 (0.40) MAPTRXFP1GRM4
SCHEMBL29028776 0.81 MPO (0.42) DYRK1AKDM4EPDE10AGRM4MAPK1
SCHEMBL29028704 0.76 MEN1 (0.45) MAPTKDM4ERXFP1PDE10AMAPK1
SCHEMBL29028803 0.76 ALDH1A1 (0.41) MAPTCLK4KDM4EPDE10AMAPK1
SCHEMBL29028680 0.72 NPC1 (0.43) MAPTKDM4EALDH1A1PDPK1NPC1
SCHEMBL29028787 0.72 MAPT (0.46) MAPTKDM4EALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332851-A Cyanomethyl phenyl indazole compound and preparation method thereof 河南中医药大学 2023-06-27 CN disclosed