SCHEMBL29424176

SCHEMBL29424176

O=C(O)Cc1ccc2oc(-c3ccc(NC(=O)/C=C/c4ccc(Br)cc4)c(F)c3)nc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20280936 1.00 HPSE (1.00) HPSE
SCHEMBL6821029 1.00 HPSE (1.00) HPSE
SCHEMBL6821869 0.94 HPSE (0.89) HPSE
SCHEMBL6821844 0.92 HPSE (1.00) HPSE
SCHEMBL6822223 0.90 HPSE (0.90) HPSE
SCHEMBL6822193 0.90 HPSE (1.00) HPSE
SCHEMBL6822288 0.89 HPSE (1.00) HPSE
SCHEMBL6824237 0.89 HPSE (1.00) HPSE
SCHEMBL7118415 0.89 HPSE (0.87) HPSE
SCHEMBL6818350 0.88 HPSE (0.83) HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 114 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637473-B2 MDM2 protein degraders REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2026-05-26 US disclosed
US-12637415-B2 Lyophilized composition comprising (s)-isopropyl 2-((s)-2-acetamido-3-(1H-indol-3-yl)propanamido)-6-diazo-5-oxohexanoate for intravenous administration and the use thereof DRACEN PHARMACEUTICALS, INC. (US) 2026-05-26 US disclosed
US-12616679-B2 Lyophilized composition comprising (s)-isopropyl 2-((s)-2-acetamido-3-(1H-indol-3-yl)propanamido)-6-diazo-5-oxohexanoate for subcutaneous administration and the use thereof DRACEN PHARMACEUTICALS, INC. (US) 2026-05-05 US disclosed
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2026-03-17 US disclosed
US-12570679-B2 STAT3 protein degraders REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2026-03-10 US disclosed
US-20260055097-A9 NRF2 PROTEIN DEGRADERS GANYMEDE ONCOLOGY INC (US) 2026-02-26 US disclosed
US-12522623-B2 Small molecule STAT protein degraders REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2026-01-13 US disclosed
US-20250295638-A1 METHODS OF TREATING ALLOGRAFT REJECTION BARGENT THERAPEUTICS PTY LTD (AU) 2025-09-25 US disclosed
US-20250276993-A1 PSEUDO-DISACCHARIDE COMPOUNDS UNIVERSITEIT LEIDEN (NL) 2025-09-04 US disclosed
US-20250215039-A1 NUCLEOSIDES FOR TREATING CANCER PRIMEFOUR THERAPEUTICS INC (US) 2025-07-03 US disclosed
EP-3569601-B1 N-(PHENYLSULFONYL)BENZAMIDES AND RELATED COMPOUNDS AS BCL-2 INHIBITORS UNIV MICHIGAN REGENTS (US) 2022-06-22 EP disclosed
US-11365186-B2 Substituted benzimidazoles, their preparation and their use as pharmaceuticals EPIGENETIX, INC. (US) 2022-06-21 US disclosed
US-20220185831-A1 STAT3 PROTEIN DEGRADERS UNIV MICHIGAN REGENTS (US) 2022-06-16 US disclosed
EP-3999510-A1 IMIDAZOPYRIMIDINES AS EED INHIBITORS AND THE USE THEREOF The Regents Of The University Of Michigan (US) 2022-05-25 EP disclosed
EP-4001273-A2 AMINOPYRIMIDINES AS ALK INHIBITORS The Regents Of The University Of Michigan (US) 2022-05-25 EP disclosed
US-20220117938-A1 COMBINATON THERAPY WITH A DON PRODRUG AND AN IMMUNE CHECKPOINT INHIBITOR DRACEN PHARMACEUTICALS, INC. 2022-04-21 US disclosed
EP-3983084-A1 AMINO ACID TRANSPORT INHIBITORS AND THE USES THEREOF Vanderbilt University (US) 2022-04-20 EP disclosed
EP-3983377-A1 DIBENZYLAMINES AS AMINO ACID TRANSPORT INHIBITORS Vanderbilt University (US) 2022-04-20 EP disclosed
WO-2022066882-A1 METHOD FOR TREATING CANCER WITH A REVERSE TRANSCRIPTASE INHIBITOR ONCOLINEA PHARMACEUTICALS, INC. (US) 2022-03-31 WO disclosed
US-11267822-B2 BET bromodomain protein degraders with cleavable linkers THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2022-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (13 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12637473-B2 MDM2 protein degraders MDM2, TP53, TP53BP1 HPSE 3730/4885
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors BCL2A1, BCL2L1, BCL2L11 HPSE 3313/4885
US-11365186-B2 Substituted benzimidazoles, their preparation and their use as pharmaceuticals BRD3, BRDT, BRD4 HPSE 3410/4885
US-11267822-B2 BET bromodomain protein degraders with cleavable linkers BRD4, BET1, BRWD1 HPSE 3059/4885
US-20220117938-A1 COMBINATON THERAPY WITH A DON PRODRUG AND AN IMMUNE CHECKPOINT INHIBITOR PDCD1, CD274, BID HPSE 2612/4885
US-20220185831-A1 STAT3 PROTEIN DEGRADERS STAT3, JAK2, STAT5A HPSE 2450/4885
US-12570679-B2 STAT3 protein degraders STAT3, JAK2, IL6ST HPSE 2433/4885
US-20250276993-A1 PSEUDO-DISACCHARIDE COMPOUNDS HPSE, HEXD, HEXA HPSE 1/4885
US-12616679-B2 Lyophilized composition comprising (s)-isopropyl 2-((s)-2-acetamido-3-(1H-indol-3-yl)propanamido)-6-diazo-5-oxohexanoate for subcutaneous administration and the use thereof GLUL, QPCT, QPCTL HPSE 4645/4885
US-20250215039-A1 NUCLEOSIDES FOR TREATING CANCER UNG, OGG1, NTPCR HPSE 1047/4885
US-20250295638-A1 METHODS OF TREATING ALLOGRAFT REJECTION CD74, TST, SERPINB1 HPSE 461/4885
US-20260055097-A9 NRF2 PROTEIN DEGRADERS KEAP1, NFE2L2, NFE2 HPSE 3229/4885
US-12637415-B2 Lyophilized composition comprising (s)-isopropyl 2-((s)-2-acetamido-3-(1H-indol-3-yl)propanamido)-6-diazo-5-oxohexanoate for intravenous administration and the use thereof GLS, GLUL, GLS2 HPSE 4627/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.