SCHEMBL29519366

SCHEMBL29519366

O=C(Nc1ccc(C(=O)O)cc1)OCCC1c2cc(Cl)ccc2-c2ccc(Cl)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G4A P47712 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
BCL2 P10415 2/20 0.42
BCL2L1 Q07817 2/20 0.42
PYGL P06737 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CHRM3 P20309 2/20 0.40
NHERF1 O14745 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
F11 P03951 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL608997 0.83 EPHX2 (0.48) SMN1; SMN2NPC1RAB9AMEN1KMT2A
SCHEMBL8993314 0.77 NPC1 (0.49) SMN1; SMN2L3MBTL1NPC1RAB9AMEN1
SCHEMBL8993272 0.76 NPC1 (0.48) SMN1; SMN2NPC1RAB9AMEN1KMT2A
SCHEMBL8993273 0.72 F11 (0.41) PYGLNHERF1F11MAPTHPGD
SCHEMBL608667 0.71 EPHX2 (0.46) SMN1; SMN2NPC1RAB9AMEN1KMT2A
SCHEMBL29561956 0.70 EPHX2 (0.63) KMT2AALDH1A1
SCHEMBL29401210 0.70 EPHX2 (0.63) KMT2AALDH1A1
SCHEMBL118052 0.70 EPHX2 (0.63) KMT2AALDH1A1
SCHEMBL3007602 0.69 CSNK2A2 (0.60) SMN1; SMN2L3MBTL1NPC1RAB9AMEN1
SCHEMBL14614384 0.68 KDM4E (0.44) PLA2G4ASMN1; SMN2BCL2BCL2L1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735446-A1 SALTS AND SOLID FORMS OF A COMPOUND THAT MODULATES IRAK4 GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
EP-4735431-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
US-20260035374-A1 PYRROLO[1,2-b]PYRIDAZINE DERIVATIVES GILEAD SCIENCES INC (US) 2026-02-05 US disclosed
EP-4674484-A2 THIENOPYRROLE COMPOUNDS Gilead Sciences, Inc. (US) 2026-01-07 EP disclosed
US-12415808-B2 Pyrrolo[1,2-b]pyridazine derivatives GILEAD SCIENCES, INC. (US) 2025-09-16 US disclosed
EP-4291562-B1 THIENOPYRROLE COMPOUNDS GILEAD SCIENCES INC (US) 2025-09-10 EP disclosed
US-12240862-B2 Inhibitors of peptidylarginine deiminases GILEAD SCIENCES, INC. (US) 2025-03-04 US disclosed
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. 2025-02-13 US disclosed
US-20250049780-A1 THIENOPYRROLE COMPOUNDS GILEAD SCIENCES, INC. 2025-02-13 US disclosed
US-20250034154-A1 SALTS AND SOLID FORMS OF A COMPOUND THAT MODULATES IRAK4 GILEAD SCIENCES, INC. 2025-01-30 US disclosed
US-20220402910-A1 THIADIAZOLE IRAK4 INHIBITORS GILEAD SCIENCES, INC. 2022-12-22 US disclosed
US-20220389034-A1 THIENOPYRROLE COMPOUNDS GILEAD SCIENCES, INC. 2022-12-08 US disclosed
WO-2022221642-A1 THIENOPYRROLE COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-10-20 WO disclosed
WO-2022173722-A1 THIENOPYRROLE COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-08-18 WO disclosed
US-20220227787-A1 INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. 2022-07-21 US disclosed
WO-2022140325-A1 6-SUBSTITUTED INDOLE COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed
WO-2022140428-A2 INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed
WO-2022140390-A1 INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed
WO-2022140326-A1 SUBSTITUTED INDOLE COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed
US-20220098187-A1 THIADIAZOLE IRAK4 INHIBITORS GILEAD SCIENCES, INC. 2022-03-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260035374-A1 PYRROLO[1,2-b]PYRIDAZINE DERIVATIVES IRAK4, IRAK1, IRAK2 PLA2G4A 1891/4885SMN1; SMN2 1133/4885L3MBTL1 1736/4885
US-20220098187-A1 THIADIAZOLE IRAK4 INHIBITORS IRAK4, IRAK3, IRAK1 PLA2G4A 3419/4885SMN1; SMN2 1294/4885L3MBTL1 780/4885
US-20250049780-A1 THIENOPYRROLE COMPOUNDS SSB, TPMT, LCP2 PLA2G4A 384/4885SMN1; SMN2 4502/4885L3MBTL1 3714/4885
US-20250034154-A1 SALTS AND SOLID FORMS OF A COMPOUND THAT MODULATES IRAK4 IRAK4, IRAK2, IRAK3 PLA2G4A 2457/4885SMN1; SMN2 2462/4885L3MBTL1 1199/4885
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME DUSP2, MKNK2, DUSP22 PLA2G4A 529/4885SMN1; SMN2 3384/4885L3MBTL1 4657/4885
US-20220227787-A1 INHIBITORS OF PEPTIDYLARGININE DEIMINASES PADI4, PADI2, PADI1 PLA2G4A 602/4885SMN1; SMN2 3144/4885L3MBTL1 3215/4885
US-20220389034-A1 THIENOPYRROLE COMPOUNDS SSB, TPMT, LCP2 PLA2G4A 384/4885SMN1; SMN2 4502/4885L3MBTL1 3714/4885
US-20220402910-A1 THIADIAZOLE IRAK4 INHIBITORS IRAK4, IRAK3, IRAK1 PLA2G4A 3419/4885SMN1; SMN2 1294/4885L3MBTL1 780/4885
US-12415808-B2 Pyrrolo[1,2-b]pyridazine derivatives CYP11B2, CYP11B1, DHPS PLA2G4A 2815/4885SMN1; SMN2 864/4885L3MBTL1 3940/4885
US-12240862-B2 Inhibitors of peptidylarginine deiminases PADI4, PADI2, PADI1 PLA2G4A 649/4885SMN1; SMN2 2054/4885L3MBTL1 2977/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.