SCHEMBL2952277

SCHEMBL2952277

Cc1nc(N2CCC(N3CCOCC3)CC2)ccc1-n1cnc2c(N)nc(N)nc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.45
HRH3 Q9Y5N1 3/20 0.41
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
AKT1 P31749 1/20 0.34
MTOR P42345 1/20 0.34
ATR Q13535 1/20 0.33
PIK3CD O00329 1/20 0.33
FLT3 P36888 1/20 0.33
CYP1A2 P05177 1/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
CXCR4 P61073 1/20 0.33
BMPR1B O00238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2953119 0.80 TTK (0.43) HRH3CYP3A4FLT3ACVR1SMPD3
SCHEMBL2952940 0.77 SMPD3 (0.41) MAP4K4HRH3PIK3CDSMPD3
SCHEMBL2955719 0.77 CTSS (0.37) ATRCDK1CCNB1CCNE1CDK2
SCHEMBL2951937 0.73 DHFR (0.45) CRHBPCRHR2MTORPIK3CDCDK1
SCHEMBL2950069 0.73 ADORA2A (0.49) MAP4K4HRH3CYP1A2CDK1CCNB1
SCHEMBL2953061 0.69 DHFR (0.42) CYP2D6CRHBPCRHR2MTORCYP1A2
SCHEMBL2952950 0.69 DHFR (0.43) MTORFLT3
SCHEMBL2955288 0.69 TLR7 (0.42) PIK3CDCDK1CCNB1CCNE1CDK2
SCHEMBL2946049 0.68 DHFR (0.42) CDK1CCNB1CCNE1CDK2
SCHEMBL2952077 0.67 INSR (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111406-A2 COMPOUNDS AND THERAPEUTIC USES THEREOF MYRIAD PHARMACEUTICALS, INC. (US) 2010-09-30 WO claimed