Vapreotide

Vapreotide

SCHEMBL29580907

CC(=O)O.CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@@H](NC(=O)[C@H](N)Cc2ccccc2)CSSC[C@@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(N)=O)NC1=O

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Vapreotide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SSTR2 known ✓ P30874 16/20 0.80
SSTR5 known ✓ P35346 15/20 0.80
SSTR3 known ✓ P32745 8/20 0.78
SSTR1 P30872 2/20 0.78
SSTR4 P31391 7/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Vapreotide SCHEMBL29384009 1.00 SSTR2 (0.80) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL294911 1.00 SSTR2 (0.80) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL30163296 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL4826 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL29405608 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL4827 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL31632623 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL6369050 0.99 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL5200070 0.97 SSTR2 (0.78) SSTR2SSTR5SSTR3SSTR1SSTR4
SCHEMBL23482743 0.97 SSTR5 (0.78) SSTR2SSTR5SSTR3SSTR1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250381290-A1 Antibody Conjugates and Methods of Making and Using the Same SCHERER TECHNOLOGIES LLC R P (US) 2025-12-18 US disclosed
US-20250262315-A1 TRIPEPTIDE LINKERS AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2025-08-21 US disclosed
EP-4592275-A2 HYDRAZINYL-PYRROLO COMPOUNDS AND METHODS FOR PRODUCING A CONJUGATE Redwood Bioscience, Inc. (US) 2025-07-30 EP disclosed
EP-3074010-B1 HYDRAZINYL-PYRROLO COMPOUNDS AND METHODS FOR PRODUCING A CONJUGATE REDWOOD BIOSCIENCE INC (US) 2025-05-14 EP disclosed
US-12296021-B2 Antibody conjugates and methods of making and using the same R.P. SCHERER TECHNOLOGIES, LLC (US) 2025-05-13 US disclosed
US-20250115546-A1 LINKERS FOR ANTIBODY DRUG CONJUGATES UNIV TEXAS (US) 2025-04-10 US disclosed
US-12215080-B2 Hydrazinyl-pyrrolo compounds and methods for producing a conjugate REDWOOD BIOSCIENCE, INC. (US) 2025-02-04 US disclosed
EP-4452292-A2 TRIPEPTIDE LINKERS AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-10-30 EP disclosed
CN-111065623-B9 Linker for antibody drug conjugates 德克萨斯州大学系统董事会 2024-10-25 CN disclosed
CN-118652192-A Linker for antibody drug conjugates 德克萨斯州大学系统董事会 2024-09-17 CN disclosed
WO-2023122587-A2 TRIPEPTIDE LINKERS AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-06-29 WO disclosed
US-11629122-B2 Linkers for antibody drug conjugates THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-04-18 US disclosed
US-20230068124-A1 Hydrazinyl-Indole Compounds and Methods for Producing a Conjugate ARES CAPITAL CORPORATION, AS COLLATERAL AGENT 2023-03-02 US disclosed
CN-115504924-A Hydrazino-pyrrolo compounds and methods for forming conjugates 雷德伍德生物科技股份有限公司 2022-12-23 CN disclosed
US-11466096-B2 Antibody conjugates and methods of making and using the same R.P. SCHERER TECHNOLOGIES, LLC (US) 2022-10-11 US disclosed
CN-105744935-B Hydrazino-pyrrolo compounds and methods for forming conjugates 雷德伍德生物科技股份有限公司 2022-09-30 CN disclosed
US-11426465-B2 Hydrazinyl-indole compounds and methods for producing a conjugate Redwiid Bioscience, Inc. (US) 2022-08-30 US disclosed
US-11376334-B2 Hydrazinyl-substituted heteroaryl compounds and methods for producing a conjugate R.P. SCHERER TECHNOLOGIES, LLC (US) 2022-07-05 US disclosed
US-20220153696-A1 Hydrazinyl-Pyrrolo Compounds and Methods for Producing a Conjugate ARES CAPITAL CORPORATION, AS COLLATERAL AGENT 2022-05-19 US disclosed
US-20220145270-A1 Antibody Conjugates and Methods of Making and Using the Same ARES CAPITAL CORPORATION, AS COLLATERAL AGENT 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230068124-A1 Hydrazinyl-Indole Compounds and Methods for Producing a Conjugate HNMT, AANAT, INMT SSTR2 628/4885SSTR5 84/4885SSTR3 445/4885
US-20220153696-A1 Hydrazinyl-Pyrrolo Compounds and Methods for Producing a Conjugate DNPEP, QPCT, PDS5A SSTR2 3008/4885SSTR5 802/4885SSTR3 2594/4885
US-20250115546-A1 LINKERS FOR ANTIBODY DRUG CONJUGATES CD47, EPCAM, SDCBP SSTR2 2302/4885SSTR5 789/4885SSTR3 2121/4885
US-11426465-B2 Hydrazinyl-indole compounds and methods for producing a conjugate HNMT, AANAT, INMT SSTR2 628/4885SSTR5 84/4885SSTR3 445/4885
US-20250381290-A1 Antibody Conjugates and Methods of Making and Using the Same PFAS, FGR, FGB SSTR2 3589/4885SSTR5 2312/4885SSTR3 2313/4885
US-20250262315-A1 TRIPEPTIDE LINKERS AND METHODS OF USE THEREOF DNPEP, VIP, LNPEP SSTR2 1545/4885SSTR5 623/4885SSTR3 607/4885
US-12215080-B2 Hydrazinyl-pyrrolo compounds and methods for producing a conjugate DNPEP, QPCT, PDS5A SSTR2 3008/4885SSTR5 802/4885SSTR3 2594/4885
US-11376334-B2 Hydrazinyl-substituted heteroaryl compounds and methods for producing a conjugate HNMT, TIAL1, HACL2 SSTR2 3211/4885SSTR5 1345/4885SSTR3 2259/4885
US-11629122-B2 Linkers for antibody drug conjugates CD47, EPCAM, FCGRT SSTR2 2082/4885SSTR5 571/4885SSTR3 1742/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.