Vapreotide

Vapreotide

SCHEMBL29405608

CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](NC(=O)[C@H](N)Cc2ccccc2)CSSC[C@@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(N)=O)NC1=O

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Vapreotide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SSTR2 known ✓ P30874 16/20 0.81
SSTR5 known ✓ P35346 15/20 0.81
SSTR3 known ✓ P32745 8/20 0.78
SSTR1 P30872 2/20 0.78
SSTR4 P31391 7/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Vapreotide SCHEMBL4827 1.00 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL6369050 1.00 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL4826 1.00 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL31632623 1.00 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL30163296 1.00 SSTR2 (0.81) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL29580907 0.99 SSTR2 (0.80) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL294911 0.99 SSTR2 (0.80) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL29384009 0.99 SSTR2 (0.80) SSTR2SSTR5SSTR3SSTR1SSTR4
Vapreotide SCHEMBL5200070 0.97 SSTR2 (0.78) SSTR2SSTR5SSTR3SSTR1SSTR4
SCHEMBL23482743 0.97 SSTR5 (0.78) SSTR2SSTR5SSTR3SSTR1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11827651-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-11-28 US claimed
US-20220270454-A1 TREATMENT OF KIDNEY DISEASES ASSOCIATED WITH ELEVATED AVP THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2022-08-25 US claimed
US-12624002-B2 Dimers for use in synthesis of peptidomimetics THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-05-12 US disclosed
EP-4095608-B1 ELECTROSTATIC IMAGE DEVELOPING TONER FUJIFILM BUSINESS INNOVATION CORP (JP) 2026-04-29 EP disclosed
US-12600699-B2 Thiosemicarbazates and uses thereof THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-04-14 US disclosed
US-12595233-B2 Thiosemicarbazates and uses thereof THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-04-07 US disclosed
US-20260070894-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2026-03-12 US disclosed
US-12486294-B2 Radioisotope labeled compound for imaging or treatment of prostate cancer SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2025-12-02 US disclosed
WO-2025233437-A1 POLYPEPTIDE COMPRISING A CAPSID PROTEIN SEQUENCE A-SPECTAR GMBH (AT) 2025-11-13 WO disclosed
EP-4647438-A1 POLYPEPTIDE COMPRISING A CAPSID PROTEIN SEQUENCE A-Spectar GmbH (AT) 2025-11-12 EP disclosed
US-12351573-B2 Compounds for use in synthesis of peptidomimetics THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH (US) 2025-07-08 US disclosed
US-11392052-B2 Electrostatic image developing toner, electrostatic image developer, toner cartridge, process cartridge, image forming apparatus, and image forming method FUJIFILM BUSINESS INNOVATION CORP. (JP) 2022-07-19 US disclosed
US-11354990-B2 Treatment of kidney diseases associated with elevated AVP THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2022-06-07 US disclosed
CN-107203103-B Image forming method and image forming apparatus 富士胶片商业创新有限公司 2022-06-03 CN disclosed
US-11324827-B2 Multifunctionalized polyethylene glycol derivative and preparation method therefor XIAMEN SINOPEG BIOTECH CO., LTD. (CN) 2022-05-10 US disclosed
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS ON TARGET THERAPEUTICS LLC 2022-05-05 US disclosed
US-20220088150-A1 Octreotide Microsphere-Based Arterial Embolization for Treating Obesity BIOVENA SCIENCE LLC (US) 2022-03-24 US disclosed
EP-3966201-A1 THIOSEMICARBAZATES AND USES THEREOF The Feinstein Institutes for Medical Research (US) 2022-03-16 EP disclosed
EP-3966223-A1 PEPTIDOMIMETIC AGENTS, SYNTHESIS AND USES THEREOF The Feinstein Institutes for Medical Research (US) 2022-03-16 EP disclosed
CN-114126619-A Compounds for the synthesis of peptidomimetics 范因斯坦医学研究院 2022-03-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12351573-B2 Compounds for use in synthesis of peptidomimetics DNPEP, NPEPPS, PAM SSTR2 62/4885SSTR5 126/4885SSTR3 79/4885
US-20220135633-A1 METHODS AND SYSTEMS FOR DESIGNING AND/OR CHARACTERIZING SOLUBLE LIPIDATED LIGAND AGENTS LDLR, HDLBP, LIPG SSTR2 2069/4885SSTR5 3066/4885SSTR3 2297/4885
US-12486294-B2 Radioisotope labeled compound for imaging or treatment of prostate cancer ARGLU1, KLK3, GLUL SSTR2 1231/4885SSTR5 517/4885SSTR3 872/4885
US-12624002-B2 Dimers for use in synthesis of peptidomimetics GLUL, ARGLU1, ASNS SSTR2 299/4885SSTR5 630/4885SSTR3 228/4885
US-11354990-B2 Treatment of kidney diseases associated with elevated AVP AVPR2, PKD1, AVPR1A SSTR2 1518/4885SSTR5 1178/4885SSTR3 1039/4885
US-20260070894-A1 COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS NPR1, NGLY1, DDAH1 SSTR2 119/4885SSTR5 68/4885SSTR3 55/4885
US-12595233-B2 Thiosemicarbazates and uses thereof TST, THRB, HSPB1 SSTR2 501/4885SSTR5 106/4885SSTR3 217/4885
US-11324827-B2 Multifunctionalized polyethylene glycol derivative and preparation method therefor HDGF, F11, F12 SSTR2 2189/4885SSTR5 2683/4885SSTR3 2107/4885
US-12600699-B2 Thiosemicarbazates and uses thereof MET, THRB, ABAT SSTR2 988/4885SSTR5 503/4885SSTR3 479/4885
US-11827651-B2 Organic electroluminescent materials and devices SSB, L1CAM, LEF1 SSTR2 2395/4885SSTR5 4107/4885SSTR3 3010/4885
US-20220270454-A1 TREATMENT OF KIDNEY DISEASES ASSOCIATED WITH ELEVATED AVP AVPR2, PKD1, AVPR1A SSTR2 1501/4885SSTR5 1145/4885SSTR3 1013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.