Sb-243213

Sb-243213

SCHEMBL29697170

Cc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1ccc(Oc3cccnc3C)nc1)CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 20/20 1.00
HTR2B P41595 19/20 1.00
HTR2A P28223 18/20 1.00
CYP2C9 P11712 1/20 1.00
HTR6 P50406 1/20 1.00
NPC1 O15118 1/20 0.77
MTOR P42345 1/20 0.77
RAB9A P51151 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sb-243213 SCHEMBL31060820 1.00 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
Sb-243213 SCHEMBL677610 1.00 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
Sb-243213 SCHEMBL18321797 0.99 HTR2C (0.98) HTR2CHTR2BHTR2ACYP2C9HTR6
Sb-243213 SCHEMBL7473195 0.99 HTR2C (0.98) HTR2CHTR2BHTR2ACYP2C9HTR6
SCHEMBL7078894 0.93 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
SCHEMBL7082914 0.90 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
SCHEMBL7473325 0.88 HTR2A (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
SCHEMBL2229787 0.87 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
Sb-242084 SCHEMBL29388888 0.87 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6
Sb-242084 SCHEMBL29462298 0.87 HTR2C (1.00) HTR2CHTR2BHTR2ACYP2C9HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 103 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000641-A1 ISOTOPICALLY ENRICHED ANALOGS OF 5,6-METHYLENEDIOXY-2-AMINOINDANE (IMDAI) TERRAN BIOSCIENCES INC (US) 2026-01-01 US claimed
US-20250136548-A1 FUNCTIONALIZED ALKYLAMINES TERRAN BIOSCIENCES INC (US) 2025-05-01 US claimed
US-20250129064-A1 PRODRUGS OF 2-BROMO-LSD (2-BROMOLYSERGIC ACID DIETHYLAMIDE) TERRAN BIOSCIENCES INC. 2025-04-24 US claimed
US-20250129054-A1 PRODRUGS OF 3,4-METHYLENEDIOXY-N-METHCATHINONE AND USES THEREOF TERRAN BIOSCIENCES INC (US) 2025-04-24 US claimed
US-20250109130-A1 ISOTOPICALLY ENRICHED ANALOGS OF 2-BROMO-LSD, LSD, ALD-52, AND 1P-LSD TERRAN BIOSCIENCES INC (US) 2025-04-03 US claimed
US-20250091993-A1 SALTS AND SOLID FORMS OF N-ETHYL-2-(5-FLUORO-1H-INDOL-3-YL)-N-METHYLETHAN-1-AMINE TERRAN BIOSCIENCES INC (US) 2025-03-20 US claimed
US-20250066299-A1 SALTS AND SOLID FORMS OF 4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE HEMI-GLUTARATE AND HEMI-SUCCINATE TERRAN BIOSCIENCES INC (US) 2025-02-27 US claimed
US-20250034105-A1 ISOTOPICALLY ENRICHED N-METHYL-1,3-BENZODIOXOLYLBUTANAMINE (MBDB) AND STEREOISOMERS THEREOF TERRAN BIOSCIENCES INC (US) 2025-01-30 US claimed
US-20250011351-A1 PSILOCYBIN AND O-ACETYLPSILOCIN, SALTS AND SOLID STATE FORMS THEREOF TERRAN BIOSCIENCES INC (US) 2025-01-09 US claimed
EP-4448518-A1 ISOTOPICALLY ENRICHED ANALOGS OF 2-BROMO-LSD, LSD, ALD-52, AND 1P-LSD Terran Biosciences Inc. (US) 2024-10-23 EP claimed
WO-2023092044-A2 PHENETHYLAMINE COMPOUNDS SALTS, POLYMORPHIC FORMS AND METHODS OF USE THEREOF TERRAN BIOSCIENCES, INC. (US) 2023-05-25 WO claimed
WO-2023086962-A1 PSILOCYBIN AND O-ACETYLPSILOCIN, SALTS AND SOLID STATE FORMS THEREOF TERRAN BIOSCIENCES INC. (US) 2023-05-19 WO claimed
WO-2023087034-A1 SALTS AND SOLID FORMS OF 4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE TERRAN BIOSCIENCES, INC. (US) 2023-05-19 WO claimed
WO-2023081899-A1 ISOTOPICALLY ENRICHED N-METHYL-1,3-BENZODIOXOLYLBUTANAMINE (MBDB) AND STEREOISOMERS THEREOF TERRAN BIOSCIENCES, INC. (US) 2023-05-11 WO claimed
WO-2023081897-A1 ISOTOPICALLY ENRICHED 3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE (MDE) AND STEREOISOMERS THEREOF TERRAN BIOSCIENCES, INC. (US) 2023-05-11 WO claimed
WO-2023081895-A1 ISOTOPICALLY ENRICHED ANALOGS OF 5,6-METHYLENEDIOXY-2-AMINOINDANE (MDAI) TERRAN BIOSCIENCES, INC. (US) 2023-05-11 WO claimed
WO-2023077127-A2 N-SUBSTITUTED INDOLES TERRAN BIOSCIENCES, INC. (US) 2023-05-04 WO claimed
WO-2023077125-A2 AZEPINO-INDOLES FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS TERRAN BIOSCIENCES, INC. (US) 2023-05-04 WO claimed
US-20220273680-A1 Methods of Treating Psychological and Brain Disorders UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-09-01 US claimed
CN-114599355-A Method for treating psychological and cerebral diseases 马里兰大学巴尔的摩分校 2022-06-07 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250129054-A1 PRODRUGS OF 3,4-METHYLENEDIOXY-N-METHCATHINONE AND USES THEREOF CYP2C19, CYP11B1, CYP2D6 HTR2C 433/4885HTR2B 489/4885HTR2A 973/4885
US-20250091993-A1 SALTS AND SOLID FORMS OF N-ETHYL-2-(5-FLUORO-1H-INDOL-3-YL)-N-METHYLETHAN-1-AMINE SLC1A2, SLC6A4, SLC6A3 HTR2C 44/4885HTR2B 397/4885HTR2A 48/4885
US-20260000641-A1 ISOTOPICALLY ENRICHED ANALOGS OF 5,6-METHYLENEDIOXY-2-AMINOINDANE (IMDAI) DRD2, HTR1D, DRD1 HTR2C 4/4885HTR2B 33/4885HTR2A 7/4885
US-20250109130-A1 ISOTOPICALLY ENRICHED ANALOGS OF 2-BROMO-LSD, LSD, ALD-52, AND 1P-LSD LMNB2, CLN6, EPM2A HTR2C 32/4885HTR2B 36/4885HTR2A 10/4885
US-20250136548-A1 FUNCTIONALIZED ALKYLAMINES BDNF, HTR2A, NTRK2 HTR2C 6/4885HTR2B 8/4885HTR2A 2/4885
US-20250011351-A1 PSILOCYBIN AND O-ACETYLPSILOCIN, SALTS AND SOLID STATE FORMS THEREOF AANAT, PSAP, SPTSSB HTR2C 604/4885HTR2B 209/4885HTR2A 493/4885
US-20250034105-A1 ISOTOPICALLY ENRICHED N-METHYL-1,3-BENZODIOXOLYLBUTANAMINE (MBDB) AND STEREOISOMERS THEREOF DBH, PNMT, MBTD1 HTR2C 208/4885HTR2B 43/4885HTR2A 341/4885
US-20250066299-A1 SALTS AND SOLID FORMS OF 4-HYDROXY-N,N-DIISOPROPYLTRYPTAMINE HEMI-GLUTARATE AND HEMI-SUCCINATE SLC6A4, SLC6A3, SLC6A2 HTR2C 60/4885HTR2B 168/4885HTR2A 91/4885
US-20250129064-A1 PRODRUGS OF 2-BROMO-LSD (2-BROMOLYSERGIC ACID DIETHYLAMIDE) GBA2, GBA1, SLC18A2 HTR2C 16/4885HTR2B 23/4885HTR2A 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.