SCHEMBL29965

SCHEMBL29965

Fc1ccccc1O[C]1CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.47
SLC6A2 P23975 7/20 0.47
SLC6A3 Q01959 4/20 0.47
SLC6A4 P31645 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ESR1 P03372 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PARP10 Q53GL7 1/20 0.43
CXCL8 P10145 1/20 0.43
RHEB Q15382 1/20 0.42
ADRB2 P07550 1/20 0.39
HSPB1 P04792 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MRGPRX1 Q96LB2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30773497 0.82 HTR1A (0.55) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL2389927 0.82 HTR1A (0.55) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL6293887 0.79 HTR1A (0.59) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL6289414 0.79 HTR1A (0.59) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL6289399 0.79 HTR1A (0.59) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL6293091 0.79 HTR1A (0.59) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL29554 0.77 HSPB1 (0.46) HSPB1
SCHEMBL6293051 0.75 PARP10 (0.66) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL702582 0.73 PARP10 (0.58) HTR1ASLC6A2SLC6A3SLC6A4ALDH1A1
SCHEMBL6289863 0.73 PARP10 (0.63) HTR1ASLC6A2SLC6A3ALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9241487-B2 Pyrimidine derivatives and use thereof as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-26 US disclosed
US-9198429-B2 Heterocyclic alkanol-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-01 US disclosed
CN-103180301-B 5-iodo triazole derivative BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-25 CN disclosed
US-9095136-B2 2-IODO imidazole-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-04 US disclosed
EP-2609088-B1 5-IODO-TRIAZOLE DERIVATIVES BAYER IP GMBH (DE) 2015-04-29 EP disclosed
US-8969248-B2 5-iodotriazole derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-03-03 US disclosed
US-20140336232-A1 2-IODO IMIDAZOLE-DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-11-13 US disclosed
CN-104066725-A Novel heterocyclic alkanol derivatives BAYER IP GMBH 2014-09-24 CN disclosed
US-20140274952-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES BAYER INTELLCTUAL PROPERTY GMBH (DE) 2014-09-18 US disclosed
CN-104039146-A 2-iodo Imidazole-derivatives BAYER IP GMBH 2014-09-10 CN disclosed
US-20140031373-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-01-30 US disclosed
CN-103391926-A Pyrimidine derivatives and use thereof as pesticides BAYER IP GMBH 2013-11-13 CN disclosed
EP-2646418-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES Bayer Intellectual Property GmbH (DE) 2013-10-09 EP disclosed
EP-2609088-A1 5-IODO-TRIAZOLE DERIVATIVES Bayer Intellectual Property GmbH (DE) 2013-07-03 EP disclosed
CN-103180301-A 5-iodo-triazole derivatives BAYER CROPSCIENCE AG 2013-06-26 CN disclosed
US-20120220638-A1 5-Iodotriazole derivatives BAYER CROPSCIENCE AG (DE) 2012-08-30 US disclosed
WO-2012072547-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-06-07 WO disclosed
WO-2012025506-A1 5-IODO-TRIAZOLE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2012-03-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140336232-A1 2-IODO IMIDAZOLE-DERIVATIVES CIP2A, ING2, AZI2 HTR1A 3848/4885SLC6A2 4614/4885SLC6A3 4423/4885
US-20140031373-A1 PYRIMIDINE DERIVATIVES AND USE THEREOF AS PESTICIDES TYMP, TYMS, UMPS HTR1A 3588/4885SLC6A2 4458/4885SLC6A3 3862/4885
US-20120220638-A1 5-Iodotriazole derivatives INMT, IGFBP5, HDHD5 HTR1A 2432/4885SLC6A2 4205/4885SLC6A3 3072/4885
US-20140274952-A1 NOVEL HETEROCYCLIC ALKANOL-DERIVATIVES ERG28, CBR3, MYB HTR1A 3543/4885SLC6A2 4853/4885SLC6A3 4812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.