SCHEMBL2997405

SCHEMBL2997405

O=P([O-])([O-])c1ccc(Oc2ccc(O)cc2)cc1.[Na+].[Na+]

nearest known ligand 0.56

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 known ✓ Q92731 1/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
ESR1 P03372 2/20 0.56
LTA4H P09960 6/20 0.48
NR1H2 P55055 1/20 0.48
BAX Q07812 1/20 0.48
PARP10 Q53GL7 1/20 0.46
KDM4E B2RXH2 1/20 0.43
MMP2 P08253 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP14 P50281 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2997696 0.87 ESR1 (0.48) MEN1KMT2AESR1ESR2KDM4E
SCHEMBL2997406 0.78 MEN1 (0.58) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL18198 0.75 ESR2 (1.00) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL249169 0.75 ESR2 (1.00) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL7811939 0.75 ESR2 (1.00) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL3175106 0.75 ESR2 (1.00) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL14148731 0.74 LTA4H (0.63) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL3829920 0.74 LTA4H (0.69) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL3832572 0.74 LTA4H (0.69) MEN1KMT2AESR1ESR2LTA4H
SCHEMBL5705485 0.74 MEN1 (0.46) MEN1KMT2AESR1ESR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100197815-A1 Polyparaphenylene Hydrocarbon Electrolyte, Manufacture Method Therefor, and Polyparaphenylene as well as Electrolyte Membrane, Catalyst Layer and Solid Polymer Fuel Cell TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2010-08-05 US disclosed
EP-1999179-A2 POLYPARAPHENYLENE HYDROCARBON ELECTROLYTE, MANUFACTURE METHOD THEREFOR, AND POLYPARAPHENYLENE AS WELL AS ELECTROLYTE MEMBRANE, CATALYST LAYER AND SOLID POLYMER FUEL CELL TOYOTA JIDOSHA KABUSHIKI KAISHA (JP) 2008-12-10 EP disclosed
WO-2007110766-A2 POLYPARAPHENYLENE HYDROCARBON ELECTROLYTE, MANUFACTURE METHOD THEREFOR, AND POLYPARAPHENYLENE AS WELL AS ELECTROLYTE MEMBRANE, CATALYST LAYER AND SOLID POLYMER FUEL CELL TOYOTA JIDOSHA KABUSHIKI KAISHA (DE) 2007-10-04 WO disclosed