SCHEMBL312769

SCHEMBL312769

Cc1cccc(S(=O)(=O)N(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.56
NPC1 O15118 3/20 0.56
TNF P01375 1/20 0.56
NOD1 Q9Y239 1/20 0.56
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
TSHR P16473 2/20 0.53
KMT2A Q03164 8/20 0.52
MEN1 O00255 7/20 0.50
ALDH1A1 P00352 5/20 0.49
TP53 P04637 1/20 0.49
HPGD P15428 1/20 0.49
GFER P55789 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
HCRTR2 O43614 1/20 0.46
LOX P28300 1/20 0.45
MAPT P10636 3/20 0.45
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163455 0.87 RAB9A (0.63) RAB9ANPC1TNFNOD1HTR2C
SCHEMBL1460044 0.84 HTR2A (0.51) RAB9ANPC1TNFNOD1HTR2A
SCHEMBL11702941 0.82 HTR2A (0.50) RAB9ANPC1TNFNOD1HTR2A
SCHEMBL11745452 0.82 HTR2A (0.50) RAB9ANPC1TNFNOD1HTR2A
SCHEMBL1940026 0.82 KMT2A (0.50) RAB9AHTR2AHTR2CTSHRKMT2A
SCHEMBL2055333 0.81 CNR2 (0.51) RAB9ANPC1TNFNOD1HTR2A
SCHEMBL2595955 0.81 ALDH1A1 (0.63) RAB9ANPC1TNFNOD1TSHR
SCHEMBL18088392 0.80 CA12 (0.67) HTR2CALDH1A1HPGDHSD17B10MAPT
SCHEMBL9860335 0.79 ALDH1A1 (0.71) RAB9ATSHRKMT2AMEN1ALDH1A1
SCHEMBL30387998 0.78 KMT2A (0.55) HTR2AHTR2CKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100422182-C Imidazopyridine derivatives as inducible NO-synthase inhibitors ALTANA PHARMA AG (DE) 2008-10-01 CN claimed
EP-1670796-B1 IMIDAZOPYRIDINE-DERIVATIVES AS INDUCIBLE NO-SYNTHASE INHIBITORS NYCOMED GMBH (DE) 2008-06-25 EP claimed
CN-1856495-A Imidazopyridine Derivatives as Inducible NO-Synthase Inhibitors ALTANA PHARMA AG (DE) 2006-11-01 CN claimed
US-20240398811-A1 PRC2 INHIBITORS FOR USE IN TREATING BLOOD DISORDERS ORIC PHARMACEUTICALS, INC. 2024-12-05 US disclosed
WO-2024015251-A1 INHIBITORS OF HPK1 AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2024-01-18 WO disclosed
US-20230303501-A1 C-ABL TYROSINE KINASE INHIBITORY COMPOUND EMBODIMENTS AND METHODS OF MAKING AND USING THE SAME THE USA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2023-09-28 US disclosed
US-20230303501-A1 C-ABL TYROSINE KINASE INHIBITORY COMPOUND EMBODIMENTS AND METHODS OF MAKING AND USING THE SAME THE USA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2023-09-28 US disclosed
US-11759462-B2 Spirocyclic compounds as tryptophan hydroxylase inhibitors ALTAVANT SCIENCES GMBH 2023-09-19 US disclosed
US-20230118795-A1 ARYL OR HETEROARYL PYRIDONE OR PYRIMIDINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF SUZHOU ZELGEN BIOPHARMACEUTICALS CO., LTD. (CN) 2023-04-20 US disclosed
WO-2022263548-A1 3-SUBSTITUTED 1H-PYRROLO[2,3-B]PYRIDINE AS GRK5 MODULATORS LEAD DISCOVERY CENTER GMBH (DE) 2022-12-22 WO disclosed
EP-4104901-A1 3-SUBSTITUTED 1H-PYRROLO[2,3-B]PYRIDINE AS GRK5 MODULATORS Lead Discovery Center GmbH (DE) 2022-12-21 EP disclosed
US-7404632-B2 Ink-jet recording ink and image forming method FUJIFILM CORPORATION (JP) 2008-07-29 US disclosed
US-7368449-B2 2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists SCHERING CORPORATION (US) 2008-05-06 US disclosed
US-7368449-B2 2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists SCHERING CORPORATION (US) 2008-05-06 US disclosed
US-20080096882-A1 PDE4 (Phosphodiesterase) inhibitors; respiratory diseases, gastrointestinal diseases, inflammation the joints, skin or eyes, cancers, or diseases of the peripheral or central nervous system BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-04-24 US disclosed
US-20080076044-A1 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production FUJIFILM CORPORATION (JP) 2008-03-27 US disclosed
US-20070191447-A1 Novel heterocyclic compound DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2007-08-16 US disclosed
CN-1856495-A Imidazopyridine Derivatives as Inducible NO-Synthase Inhibitors ALTANA PHARMA AG (DE) 2006-11-01 CN disclosed
US-20040220194-A1 2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists SCHERING CORPORATION 2004-11-04 US disclosed
US-20040220194-A1 2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists SCHERING CORPORATION 2004-11-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303501-A1 C-ABL TYROSINE KINASE INHIBITORY COMPOUND EMBODIMENTS AND METHODS OF MAKING AND USING THE SAME ABL1, ABL2, MUSK RAB9A 775/4885NPC1 4021/4885TNF 4076/4885
US-20070191447-A1 Novel heterocyclic compound OPRD1, GRIN3A, GRM3 RAB9A 1737/4885NPC1 1846/4885TNF 4274/4885
US-20080096882-A1 PDE4 (Phosphodiesterase) inhibitors; respiratory diseases, gastrointestinal diseases, inflammation the joints, skin or eyes, cancers, or diseases of the peripheral or central nervous system PDE4A, PDE4B, PDE12 RAB9A 2130/4885NPC1 4397/4885TNF 295/4885
US-20040220194-A1 2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists ADORA2A, ADORA3, ADORA1 RAB9A 595/4885NPC1 739/4885TNF 4769/4885
US-11759462-B2 Spirocyclic compounds as tryptophan hydroxylase inhibitors TPH1, TPH2, HTR1A RAB9A 2533/4885NPC1 2072/4885TNF 1137/4885
US-20240398811-A1 PRC2 INHIBITORS FOR USE IN TREATING BLOOD DISORDERS EZH2, BMI1, EZH1 RAB9A 921/4885NPC1 2100/4885TNF 4809/4885
US-20080076044-A1 Compound or its tautomer, metal complex compound, colored photosensitive curing composition, color filter, and production PBRM1, CRY1, MAPT RAB9A 1490/4885NPC1 3836/4885TNF 2167/4885
US-20230118795-A1 ARYL OR HETEROARYL PYRIDONE OR PYRIMIDINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF KRAS, NRAS, HRAS RAB9A 151/4885NPC1 2518/4885TNF 4828/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.