SCHEMBL3264173

SCHEMBL3264173

C=CCc1oc2ccccc2c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.46
GAA P10253 5/20 0.46
ALDH1A1 P00352 4/20 0.46
MAPT P10636 6/20 0.39
KMT2A Q03164 4/20 0.39
NPC1 O15118 3/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA9 Q16790 2/20 0.39
AHR P35869 1/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 3/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NQO1 P15559 1/20 0.38
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4250447 0.79 CA12 (0.39) KDM4EALDH1A1MAPTKMT2ANPC1
SCHEMBL3988877 0.77 GAA (0.57) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL5960702 0.77 SLC22A12 (0.40) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL5694518 0.76 KDM4E (0.45) KDM4EALDH1A1MAPTKMT2ANPC1
SCHEMBL11883140 0.76 CA12 (0.37) KDM4EALDH1A1MAPTKMT2ANPC1
SCHEMBL4430343 0.75 EYA3 (0.44) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL7192591 0.73 GAA (0.57) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL13948285 0.73 PTPN1 (0.53) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL11881929 0.72 MGAM (0.35) KDM4EGAAALDH1A1MAPTKMT2A
SCHEMBL9605230 0.72 EYA3 (0.43) ALDH1A1MAPTKMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 57 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230183199-A1 2-AMINOINDANE COMPOUNDS FOR MENTAL DISORDERS OR ENHANCEMENT TACTOGEN INC. (US) 2023-06-15 US disclosed
EP-4192447-A1 2-AMINOINDANE COMPOUNDS FOR MENTAL DISORDERS OR ENHANCEMENT Tactogen Inc. (US) 2023-06-14 EP disclosed
CN-116209657-A 2-aminoindane compounds for mental disorders or enhancement 泰科根公司 2023-06-02 CN disclosed
CN-116075300-A Advantageous benzofuran compositions for mental disorders or mental enhancement 泰科根公司 2023-05-05 CN disclosed
EP-2108649-B1 Novel indol carboxylic acid bispyridyl carboxamide derivatives as 5-HT2c receptor antagonists KOREA RES INST CHEM TECH (KR) 2013-04-24 EP disclosed
US-8324246-B2 Indol carboxylic acid bispyridyl carboxamide derivatives, pharmaceutically acceptable salt thereof, preparation method and composition containing the same as an active ingredient KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2012-12-04 US disclosed
EP-1335907-B1 PIPERAZINYLPYRAZINE COMPOUNDS AS AGONIST OR ANTAGONIST OF SEROTONIN 5HT-2 RECEPTOR BIOVITRUM AB PUBL (SE) 2010-06-09 EP disclosed
EP-1513831-B1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB PUBL (SE) 2010-01-06 EP disclosed
US-20090258876-A1 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-10-15 US disclosed
WO-2009125923-A2 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA RESERACH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-10-15 WO disclosed
WO-2003000663-A1 5-HT RECEPTOR LIGANDS AND USES THEREOF PFIZER PRODUCTS INC. (US) 2003-01-03 WO disclosed
US-20020147200-A1 Novel compounds and their use PROXIMAGEN NEUROSCIENCE PLC (GB) 2002-10-10 US disclosed
US-20020103204-A1 Novel compounds and their use PROXIMAGEN NEUROSCIENCE PLC (GB) 2002-08-01 US disclosed
WO-2002040456-A1 PIPERAZINYLPYRAZINE COMPOUNDS AS AGONIST OR ANTAGONIST OF SEROTONIN 5HT-2 RECEPTOR BIOVITRUM AB (SE) 2002-05-23 WO disclosed
WO-2002040457-A1 PIPERAZINYLPYRAZINES COMPOUNDS AS ANTAGONISTS OF SEROTONIN 5-HT2 RECEPTOR BIOVITRUM AB (SE) 2002-05-23 WO disclosed
EP-1149085-A1 AMINOALKYLBENZOFURANS AS SEROTONIN (5-HT(2C)) AGONISTS ELI LILLY AND COMPANY (US) 2001-10-31 EP disclosed
EP-1149085-A1 AMINOALKYLBENZOFURANS AS SEROTONIN (5-HT(2C)) AGONISTS ELI LILLY AND COMPANY (US) 2001-10-31 EP disclosed
WO-2000044737-A1 AMINOALKYLBENZOFURANS AS SEROTONIN (5-HT(2C)) AGONISTS ELI LILLY AND COMPANY (US) 2000-08-03 WO disclosed
WO-2000044737-A1 AMINOALKYLBENZOFURANS AS SEROTONIN (5-HT(2C)) AGONISTS ELI LILLY AND COMPANY (US) 2000-08-03 WO disclosed
EP-0029311-B1 AMINOALKYL BENZOFURAN DERIVATIVES, THEIR PRODUCTION AND COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1985-01-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230183199-A1 2-AMINOINDANE COMPOUNDS FOR MENTAL DISORDERS OR ENHANCEMENT AADAT, SLC1A2, TPH2 KDM4E 3126/4885GAA 3415/4885ALDH1A1 643/4885
US-20020103204-A1 Novel compounds and their use HTR2C, HTR1A, HTR1B KDM4E 2610/4885GAA 4690/4885ALDH1A1 500/4885
US-20090258876-A1 NOVEL INDOL CARBOXYLIC ACID BISPYRIDYL CARBOXAMIDE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD AND COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT HTR2C, HTR5A, HTR2A KDM4E 1130/4885GAA 3399/4885ALDH1A1 1218/4885
US-20020147200-A1 Novel compounds and their use BRIX1, UGT1A1, NR5A1 KDM4E 1971/4885GAA 844/4885ALDH1A1 288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.