SCHEMBL3574242

SCHEMBL3574242

Cc1nc(N)c(Cl)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.37
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
GFER P55789 1/20 0.35
HSP90AA1 P07900 2/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
CENPE Q02224 3/20 0.34
TRPV1 Q8NER1 1/20 0.33
PDK1 Q15118 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
CSNK1D P48730 1/20 0.33
C5AR1 P21730 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958598 0.92 CYP2C19 (0.36) CYP2C19GAAHTTGFERHSP90AA1
SCHEMBL3574241 0.81 MLYCD (0.35) CYP2C19GAAHTTGFERCENPE
SCHEMBL9957726 0.80 MLYCD (0.34) CYP2C19GAAHTTGFERCENPE
SCHEMBL9958596 0.79 MLYCD (0.33) CYP2C19GAAHTTGFEROPRM1
SCHEMBL3574238 0.78 MLYCD (0.35) CYP2C19HSP90AA1OPRM1OPRD1CENPE
SCHEMBL3580029 0.77 MLYCD (0.34) CYP2C19HSP90AA1OPRM1OPRD1CENPE
SCHEMBL3578664 0.77 CYP2C19 (0.39) CYP2C19HSP90AA1OPRM1OPRD1CENPE
SCHEMBL3584062 0.76 GBA1 (0.34) HSP90AA1OPRM1OPRD1CENPETRPV1
SCHEMBL3576622 0.75 LMNA (0.37) HSP90AA1OPRM1OPRD1CENPETRPV1
SCHEMBL1397660 0.75 TRPM8 (0.36) OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed