SCHEMBL9958598

SCHEMBL9958598

Cc1nc(N)c(Br)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C(F)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.36
CENPE Q02224 7/20 0.35
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
GFER P55789 1/20 0.34
HSP90AA1 P07900 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
C5AR1 P21730 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574242 0.92 CYP2C19 (0.37) CYP2C19CENPEGAAHTTGFER
SCHEMBL9958596 0.82 MLYCD (0.33) CYP2C19CENPEGAAHTTGFER
SCHEMBL3574241 0.79 MLYCD (0.35) CYP2C19CENPEGAAHTTGFER
SCHEMBL9957726 0.78 MLYCD (0.34) CYP2C19CENPEGAAHTTGFER
SCHEMBL3584062 0.77 GBA1 (0.34) CENPEHSP90AA1OPRM1OPRD1
SCHEMBL3574238 0.76 MLYCD (0.35) CYP2C19CENPEHSP90AA1OPRM1OPRD1
SCHEMBL3580029 0.75 MLYCD (0.34) CYP2C19CENPEHSP90AA1OPRM1OPRD1
SCHEMBL3578664 0.75 CYP2C19 (0.39) CYP2C19CENPEHSP90AA1OPRM1OPRD1
SCHEMBL3576622 0.73 LMNA (0.37) CENPEHSP90AA1OPRM1OPRD1C5AR1
SCHEMBL3579944 0.71 MCHR1 (0.39) OPRM1OPRD1C5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed