SCHEMBL3601694

SCHEMBL3601694

COc1ccccc1Cn1cnc(-c2ccc(Cl)cc2Cl)c1C(C)N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2L2 Q92843 1/20 0.45
YTHDC1 Q96MU7 1/20 0.44
DPP4 P27487 2/20 0.43
P2RX7 Q99572 1/20 0.43
TAAR1 Q96RJ0 2/20 0.41
ADORA2A P29274 1/20 0.39
KDM4E B2RXH2 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3605612 0.88 CNR1 (0.43) DPP4P2RX7CYP1A2CYP3A4CYP2D6
SCHEMBL3605710 0.88 MEN1 (0.40) DPP4KDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL3602324 0.86 CYP11B1 (0.41) DPP4P2RX7KDM4ETP53ALDH1A1
SCHEMBL3089977 0.84 BCL2L2 (0.50) BCL2L2YTHDC1DPP4P2RX7TAAR1
SCHEMBL3593028 0.83 ALDH1A1 (0.44) DPP4TP53CYP3A4CYP2C19ALDH1A1
SCHEMBL3596602 0.83 TTR (0.40) YTHDC1DPP4SMN1; SMN2
SCHEMBL3597074 0.83 CNR1 (0.44) DPP4P2RX7TP53CYP1A2CYP3A4
SCHEMBL3598037 0.82 CXCR2 (0.47) DPP4TP53CYP3A4MAPK1ALDH1A1
SCHEMBL3595008 0.80 CXCR2 (0.50) YTHDC1DPP4P2RX7TAAR1ADORA2A
SCHEMBL3599723 0.80 CNR1 (0.42) DPP4TAAR1TP53CYP3A4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed