SCHEMBL3605710

SCHEMBL3605710

COc1ccc(Cn2cnc(-c3ccc(Cl)cc3Cl)c2[C@H](C)N)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
NR3C2 P08235 1/20 0.39
CYP3A4 P08684 4/20 0.39
CYP1A2 P05177 3/20 0.39
CYP2D6 P10635 3/20 0.39
TSHR P16473 3/20 0.39
CYP2C19 P33261 3/20 0.39
MAPK1 P28482 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
DPP4 P27487 7/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CXCR2 P25025 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3601694 0.88 BCL2L2 (0.45) CYP3A4CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL3598037 0.86 CXCR2 (0.47) MEN1KMT2AHSP90AA1HSP90AB1CYP3A4
SCHEMBL3595101 0.85 DPP4 (0.43) MEN1KMT2AHSP90AA1HSP90AB1NR3C2
SCHEMBL3595008 0.83 CXCR2 (0.50) TSHRDPP4HSD17B10CXCR2MAPT
SCHEMBL3596602 0.82 TTR (0.40) MEN1KMT2ADPP4CXCR2CNR1
SCHEMBL3605612 0.80 CNR1 (0.43) CYP3A4CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL3597074 0.79 CNR1 (0.44) CYP3A4CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL3602324 0.78 CYP11B1 (0.41) MEN1KMT2ADPP4ALDH1A1KDM4E
SCHEMBL3593028 0.77 ALDH1A1 (0.44) CYP3A4CYP2C19DPP4ALDH1A1CXCR2
SCHEMBL3600972 0.76 DPP4 (0.41) MEN1KMT2ACYP3A4CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed