SCHEMBL367747

SCHEMBL367747

CS(=O)(=O)c1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 8/20 0.48
EGFR P00533 1/20 0.42
AKR1C3 P42330 1/20 0.40
AKR1C1 Q04828 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367707 0.89 EGFR (0.44) AGTR1EGFRPTGDR2MEN1KMT2A
SCHEMBL365648 0.86 CA9 (0.45) AGTR1EGFRAKR1C3AKR1C1
SCHEMBL365826 0.85 KMT2A (0.48) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL366462 0.85 LMNA (0.46) AGTR1EGFRKDM4EALDH1A1MEN1
SCHEMBL365147 0.81 AGTR1 (0.39) AGTR1EGFRAKR1C3AKR1C1KDM4E
SCHEMBL366133 0.80 AGTR1 (0.41) AGTR1
SCHEMBL367746 0.78 EGFR (0.43) AGTR1EGFRKDM4EALDH1A1MEN1
SCHEMBL366784 0.78 SCN9A (0.50) AGTR1EGFR
SCHEMBL365722 0.77 PTGDR2 (0.35) AGTR1PTGDR2KDM4EALDH1A1MEN1
SCHEMBL365935 0.77 KDM4E (0.47) AGTR1EGFRKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed