SCHEMBL366828

SCHEMBL366828

CN(C)C(=O)Oc1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.46
ALDH1A1 P00352 1/20 0.46
KMT2A Q03164 1/20 0.46
RAB9A P51151 3/20 0.45
EGFR P00533 2/20 0.39
SRC P12931 1/20 0.39
NCEH1 Q6PIU2 5/20 0.39
LMNA P02545 2/20 0.38
NPC1 O15118 2/20 0.38
TSHR P16473 1/20 0.38
TSPO P30536 1/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367283 0.89 RAB9A (0.44) PKMALDH1A1KMT2ARAB9AEGFR
SCHEMBL364802 0.84 KDM4E (0.49) PKMALDH1A1KMT2ARAB9ALMNA
SCHEMBL365014 0.82 KDM4E (0.48) ALDH1A1KMT2AEGFRGAANPSR1
SCHEMBL366406 0.81 GABRP (0.41) PKMALDH1A1KMT2ARAB9AEGFR
SCHEMBL365213 0.81 PKM (0.39) PKMALDH1A1KMT2ARAB9AEGFR
SCHEMBL366827 0.80 KMT2A (0.45) PKMALDH1A1KMT2ARAB9ASRC
SCHEMBL365640 0.80 KMT2A (0.43) PKMALDH1A1KMT2ARAB9AEGFR
SCHEMBL367734 0.79 ATM (0.40) PKMALDH1A1KMT2ARAB9ANCEH1
SCHEMBL367205 0.77 EGFR (0.45) ALDH1A1KMT2AEGFRSRC
SCHEMBL364207 0.76 EGFR (0.47) ALDH1A1KMT2ARAB9AEGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed