SCHEMBL366900

SCHEMBL366900

CC(C)Oc1ccc(CCOc2cc(OC(=O)N(C)C)cn3c2c(C(=O)O)c2ccccc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 3/20 0.39
PLA2G4A P47712 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PABPC1 P11940 1/20 0.35
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
GCK P35557 1/20 0.34
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
ALPG P10696 1/20 0.33
PKM P14618 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ACHE P22303 2/20 0.33
SRD5A1 P18405 1/20 0.33
SRD5A2 P31213 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365915 0.93 S1PR3 (0.37) S1PR3PLA2G4ANPC1RAB9APABPC1
SCHEMBL365189 0.91 ACHE (0.37) S1PR3ACHECNR2
SCHEMBL366851 0.90 ALDH1A1 (0.38) S1PR3PLA2G4ACNR2
SCHEMBL366612 0.84 ACHE (0.38) S1PR3ACHE
SCHEMBL366751 0.84 PPARG (0.33) S1PR3ITGB1ITGA4CNR2
SCHEMBL365169 0.83 ACHE (0.41) ACHE
SCHEMBL365006 0.83 LTB4R (0.35) S1PR3NPC1RAB9AACHE
SCHEMBL366374 0.82 ALDH1A1 (0.38) PLA2G4AACHECNR2
SCHEMBL365769 0.81 LTB4R (0.39) S1PR3ITGB1ITGA4PKMCNR2
SCHEMBL366899 0.80 PLA2G4A (0.36) S1PR3PLA2G4ANPC1RAB9APABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed