SCHEMBL365147

SCHEMBL365147

O=C(O)c1c2ccccc2n2cc(S(=O)(=O)C3CC3)ccc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.39
AKR1C3 P42330 1/20 0.37
AKR1C1 Q04828 1/20 0.37
EGFR P00533 1/20 0.36
HTR2A P28223 3/20 0.35
SPR P35270 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
HTR2C P28335 2/20 0.34
KCNH2 Q12809 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR3A P46098 1/20 0.34
IDO1 P14902 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366741 0.90 EGFR (0.38) AGTR1AKR1C3AKR1C1EGFRHTR2A
SCHEMBL365648 0.81 CA9 (0.45) AGTR1AKR1C3AKR1C1EGFR
SCHEMBL367747 0.81 AGTR1 (0.48) AGTR1AKR1C3AKR1C1EGFRKDM4E
SCHEMBL365146 0.80 IDO1 (0.40) AGTR1AKR1C3EGFRHTR2ASPR
SCHEMBL366462 0.78 LMNA (0.46) AGTR1EGFRKDM4EALDH1A1MEN1
SCHEMBL366926 0.77 ALDH1A1 (0.36) EGFRHTR2AKDM4EALDH1A1HPGD
SCHEMBL366133 0.73 AGTR1 (0.41) AGTR1
SCHEMBL365935 0.73 KDM4E (0.47) AGTR1EGFRKDM4EALDH1A1POLB
SCHEMBL366888 0.73 EGFR (0.44) AGTR1EGFRKDM4EALDH1A1POLB
SCHEMBL364653 0.71 CA2 (0.43) AGTR1EGFRHTR2AALDH1A1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed