SCHEMBL365648

SCHEMBL365648

NS(=O)(=O)c1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 8/20 0.45
CA1 P00915 7/20 0.45
CA2 P00918 7/20 0.45
CA12 O43570 6/20 0.45
AGTR1 P30556 9/20 0.44
EGFR P00533 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
STAT6 P42226 1/20 0.41
HIF1A Q16665 1/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C1 Q04828 1/20 0.40
CA3 P07451 1/20 0.40
CA6 P23280 1/20 0.40
CYP2C19 P33261 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367747 0.86 AGTR1 (0.48) AGTR1EGFRAKR1C3AKR1C1
SCHEMBL365427 0.84 ALDH1A1 (0.48) CA9CA1CA2CA12CA5A
SCHEMBL366462 0.82 LMNA (0.46) AGTR1EGFR
SCHEMBL365147 0.81 AGTR1 (0.39) AGTR1EGFRAKR1C3AKR1C1
SCHEMBL366104 0.81 CA9 (0.46) CA9CA1CA2CA12CYP1A2
SCHEMBL365647 0.78 IDO1 (0.43) CA9CA1CA2CA12AGTR1
SCHEMBL366133 0.77 AGTR1 (0.41) AGTR1
SCHEMBL366888 0.77 EGFR (0.44) AGTR1EGFRCYP1A2CYP2C19
SCHEMBL365935 0.77 KDM4E (0.47) AGTR1EGFRCYP1A2CYP3A4CYP2C19
SCHEMBL367707 0.77 EGFR (0.44) AGTR1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed