SCHEMBL377365

SCHEMBL377365

CC(C)(C)P(C(C)(C)C)C1(C)CC1(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRM1 P35372 2/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
GRIN1 Q05586 1/20 0.34
KCNH2 Q12809 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
ALDH1A1 P00352 2/20 0.33
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5082418 0.78 MEN1 (0.42) MEN1KMT2AOPRM1GRIN2DGRIN3B
SCHEMBL24337423 0.75 HTR2A (0.43) KCNH2
SCHEMBL5082415 0.73 MEN1 (0.39) MEN1KMT2AOPRM1ALDH1A1OPRK1
SCHEMBL377463 0.68 MEN1 (0.35) MEN1KMT2AOPRL1
SCHEMBL6263640 0.67 MEN1 (0.40) MEN1KMT2AOPRM1GRIN2DGRIN3B
SCHEMBL3310454 0.66 MEN1 (0.46) MEN1KMT2AOPRM1GRIN2DGRIN3B
SCHEMBL5078420 0.66 MEN1 (0.46) MEN1KMT2AOPRM1GRIN2DGRIN3B
SCHEMBL5080028 0.66 MEN1 (0.46) MEN1KMT2AOPRM1GRIN2DGRIN3B
SCHEMBL9541911 0.66 MEN1 (0.46) MEN1KMT2AGRIN2DGRIN3BGRIN1
SCHEMBL11040986 0.64 MEN1 (0.44) MEN1KMT2AOPRM1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 549 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4634171-A1 PROCESS FOR THE PREPARATION OF A QUINAZOLINONE DERIVATIVE F. Hoffmann-La Roche AG (CH) 2025-10-22 EP claimed
US-20250313551-A1 PROCESS FOR THE PREPARATION OF A QUINAZOLINONE DERIVATIVE HOFFMANN-LA ROCHE INC. (US) 2025-10-09 US claimed
EP-4585268-A2 SOLID FORMS OF ISOQUINOLINONE DERIVATIVES, PROCESS OF MAKING, COMPOSITIONS COMPRISING, AND METHODS OF USING THE SAME Twelve Therapeutics, Inc. (US) 2025-07-16 EP claimed
US-12122788-B2 Process of making CFTR modulators VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-10-22 US claimed
CN-118530144-A Paen Jia preparation method of beach 中国医学科学院药物研究所 2024-08-23 CN claimed
WO-2024126634-A1 PROCESS FOR THE PREPARATION OF A QUINAZOLINONE DERIVATIVE F. HOFFMANN-LA ROCHE AG (CH) 2024-06-20 WO claimed
US-11939333-B2 Solid forms of isoquinolinones, and process of making, composition comprising, and methods of using the same INFINITY PHARMACEUTICALS, INC. (US) 2024-03-26 US claimed
US-20230399343-A1 PROCESS OF MAKING CFTR MODULATORS VERTEX PHARMACEUTICALS (SAN DIEGO) LLC 2023-12-14 US claimed
CN-114075257-B Method for preparing arylamine compound from On-DNA aryl halide 成都先导药物开发股份有限公司 2023-08-22 CN claimed
CN-116368134-A Methods of making ubiquitin JAK inhibitors and related intermediate compounds 施万生物制药研发IP有限责任公司 2023-06-30 CN claimed
CN-116253606-A Preparation method of aryl difluoromethyl alkyl sulfonyl fluoride compound 上海应用技术大学 2023-06-13 CN claimed
US-20220135576-A1 SOLID FORMS OF ISOQUINOLINONES, AND PROCESS OF MAKING, COMPOSITION COMPRISING, AND METHODS OF USING THE SAME TWELVE THERAPEUTICS, INC. 2022-05-05 US claimed
CN-112094165-A Method for preparing biaryl compound by Suzuki coupling reaction 浙江省化工研究院有限公司 2020-12-18 CN claimed
US-9233922-B2 Process for producing N-(hetero)arylazoles TAKASAGO INTERNATIONAL CORPORATION (JP) 2016-01-12 US claimed
WO-2012098044-A1 PROCESS FOR THE PREPARATION OF N,N-DIISOPROPYL-3-(2-HYDROXY-5-METHYLPHENYL)- 3-PHENYL PROPYLAMINE AND ITS SALTS STARTING FROM A NOVEL INTERMEDIATE CAMBREX PROFARMACO MILANO S.R.L. (IT) 2012-07-26 WO claimed
EP-2476665-A1 Process for the preparation of N,N-diisopropyl-3-(2-hydroxy-5-methylphenyl)- 3-phenyl propylamine and its salts starting from a novel intermediate Cambrex Profarmaco Milano S.r.l. (IT) 2012-07-18 EP claimed
US-20260148808-A1 SYSTEM AND METHOD FOR OPTIMIZING CHEMICAL REACTIONS USING MACHINE LEARNING MERCK PATENT GMBH (DE) 2026-05-28 US disclosed
US-12630496-B2 Organic compound, light-emitting device, light-emitting apparatus, electronic device, and lighting device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2026-05-19 US disclosed
EP-1592698-A2 PHOSPHINE COMPOUND, INTERMEDIATE, PALLADIUM-COMPLEX, AND USE THEREOF Takasago International Corporation (JP) 2005-11-09 EP disclosed
WO-2004072088-A2 PHOSPHINE COMPOUND, INTERMEDIATE, PALLADIUM-COMPLEX, AND USE THEREOF TAKASAGO INTERNATIONAL CORPORATION (JP) 2004-08-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230399343-A1 PROCESS OF MAKING CFTR MODULATORS CFTR, SLC26A4, TMEM109 MEN1 2440/4885KMT2A 4522/4885OPRM1 1193/4885
US-20260148808-A1 SYSTEM AND METHOD FOR OPTIMIZING CHEMICAL REACTIONS USING MACHINE LEARNING KIT, ALK, ACHE MEN1 3621/4885KMT2A 273/4885OPRM1 1455/4885
US-20220135576-A1 SOLID FORMS OF ISOQUINOLINONES, AND PROCESS OF MAKING, COMPOSITION COMPRISING, AND METHODS OF USING THE SAME PIK3CA, PIK3C2A, PIK3CD MEN1 3126/4885KMT2A 2333/4885OPRM1 2625/4885
US-11939333-B2 Solid forms of isoquinolinones, and process of making, composition comprising, and methods of using the same PIK3CA, PIK3C2A, PIK3CD MEN1 3126/4885KMT2A 2333/4885OPRM1 2625/4885
US-12122788-B2 Process of making CFTR modulators CFTR, SLC26A4, TMEM109 MEN1 2440/4885KMT2A 4522/4885OPRM1 1193/4885
US-20250313551-A1 PROCESS FOR THE PREPARATION OF A QUINAZOLINONE DERIVATIVE NQO2, SDHA, NDUFS3 MEN1 3994/4885KMT2A 1193/4885OPRM1 1746/4885
US-12630496-B2 Organic compound, light-emitting device, light-emitting apparatus, electronic device, and lighting device CRY1, NR1I2, GNA11 MEN1 1976/4885KMT2A 3569/4885OPRM1 995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.