SCHEMBL3781431

SCHEMBL3781431

CCOc1nc(NCc2ccc(F)cc2)c2nc(-c3ccc(F)cc3)nnc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.42
ERBB2 P04626 2/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP3A4 P08684 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CACNA2D1 P54289 1/20 0.39
PTGS2 P35354 3/20 0.39
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
TP53 P04637 1/20 0.37
USP1 O94782 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3791356 0.91 PTPN7 (0.40) EGFRERBB2MEN1KMT2AMAPT
SCHEMBL3785492 0.90 CTSL (0.41) EGFRERBB2MEN1KMT2AMAPT
SCHEMBL3778147 0.89 CNR2 (0.42) EGFRMEN1KMT2AMAPTLMNA
SCHEMBL3789880 0.83 LMNA (0.45) EGFRMEN1KMT2AMAPTLMNA
SCHEMBL3787119 0.81 KCNH3 (0.39) EGFRERBB2MEN1KMT2AMAPT
SCHEMBL3704729 0.79 CNR2 (0.39) CYP1A2HTT
SCHEMBL3786275 0.79 USP10 (0.47) EGFRERBB2MEN1KMT2AMAPT
SCHEMBL3782046 0.76 MPO (0.45) MEN1KMT2AMAPTLMNAGAA
SCHEMBL13286377 0.75 CNR2 (0.51) EGFRMEN1KMT2AMAPTLMNA
SCHEMBL3783407 0.74 CA1 (0.42) MAPTGAAPTGS2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed