SCHEMBL4039621

SCHEMBL4039621

Cc1cc(NC(=O)[C@H](C[C@@H](O)[CH]Cc2ccccc2)C(N)=O)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 8/20 0.46
CDK2 P24941 8/20 0.46
CCNA1 P78396 8/20 0.46
CDK7 P50613 1/20 0.39
CCNH P51946 1/20 0.39
MNAT1 P51948 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ATM Q13315 1/20 0.37
MME P08473 1/20 0.37
GAA P10253 1/20 0.35
RET P07949 2/20 0.35
AURKB Q96GD4 1/20 0.35
JAK2 O60674 1/20 0.35
NPY5R Q15761 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042233 0.82 PKM (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL4040058 0.82 ALDH1A1 (0.45) NPC1RAB9ASMN1; SMN2GAAAURKB
SCHEMBL4046147 0.79 TSHR (0.44) NPC1RAB9ASMN1; SMN2GAA
SCHEMBL4039656 0.79 HDAC1 (0.42) GAA
SCHEMBL4045052 0.76 LMNA (0.46) SMN1; SMN2ATMJAK2
SCHEMBL4044987 0.74 MMP8 (0.51) GAA
SCHEMBL4043128 0.74 PKM (0.48) NPC1RAB9ASMN1; SMN2GAA
SCHEMBL4041195 0.73 MMP1 (0.41) MME
SCHEMBL4040963 0.72 REN (0.47)
SCHEMBL3936972 0.72 REN (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651592-B1 NOVEL DIBENZO[B,F]OXEPINE-10-CARBOXAMIDES AND PHARMACEUTICAL USES THEREOF NOVARTIS AG (CH) 2009-04-29 EP disclosed