SCHEMBL4040779

SCHEMBL4040779

Cc1c(OC(=O)NC(CC2CC2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2ccc[n+]([O-])c2)oc2ccccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.34
CTSL P07711 2/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.31
MMP8 P22894 2/20 0.31
MMP3 P08254 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
GAA P10253 2/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043622 0.93 CTSK (0.39) CTSVCTSLCTSSCTSKL3MBTL1
SCHEMBL4045411 0.93 PREP (0.33) CTSKL3MBTL1ALDH1A1KDM4ECA12
SCHEMBL4040797 0.91 CTSV (0.33) CTSVCTSLCTSSCTSKL3MBTL1
SCHEMBL4046064 0.90 SMN1; SMN2 (0.35) CTSSCTSKL3MBTL1ALDH1A1KDM4E
SCHEMBL4046671 0.86 CTSK (0.41) CTSVCTSLCTSSCTSK
SCHEMBL4041817 0.83 CTSL (0.33) CTSVCTSLCTSSCTSK
SCHEMBL4047097 0.83 CTSL (0.33) CTSVCTSLCTSSCTSKSMN1; SMN2
SCHEMBL4043854 0.83 CTSK (0.39) CTSVCTSLCTSSCTSKL3MBTL1
SCHEMBL4040960 0.83 PREP (0.32) CTSKL3MBTL1KDM4ESMN1; SMN2CYP3A4
SCHEMBL4042994 0.82 CTSS (0.35) CTSVCTSLCTSSCTSKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed