SCHEMBL4043292

SCHEMBL4043292

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
RAB9A P51151 3/20 0.32
NR2F2 P24468 2/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
CHRM5 P08912 3/20 0.32
KDM4E B2RXH2 1/20 0.32
TNF P01375 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
NOD1 Q9Y239 1/20 0.32
ALOX5 P09917 1/20 0.32
CHRM1 P11229 1/20 0.32
P2RY12 Q9H244 1/20 0.32
MMP1 P03956 4/20 0.31
ADAM17 P78536 3/20 0.31
MMP13 P45452 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045853 0.93 CTSK (0.38) ALDH1A1RAB9ACTSK
SCHEMBL4045249 0.91 CTSK (0.36) LMNAP2RY12CTSK
SCHEMBL4046989 0.91 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4048186 0.90 ALDH1A1 (0.36) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4046799 0.88 ALDH1A1 (0.39) ALDH1A1PREPFAPCTSK
SCHEMBL4044695 0.86 CTSK (0.36) P2RY12MMP1ADAM17MMP13CTSK
SCHEMBL4043678 0.85 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4039771 0.85 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4048294 0.85 ALDH1A1 (0.37) ALDH1A1CHRM5LMNAMAPT
SCHEMBL4049444 0.84 PREP (0.33) PREPFAPP2RY12CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed