SCHEMBL4046989

SCHEMBL4046989

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
ELOVL6 Q9H5J4 1/20 0.37
TSHR P16473 2/20 0.36
KCNQ1 P51787 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
PREP P48147 1/20 0.34
FAP Q12884 1/20 0.34
LMNA P02545 3/20 0.34
CHRM1 P11229 1/20 0.34
GAA P10253 1/20 0.34
GFER P55789 1/20 0.34
MAPT P10636 2/20 0.33
NR2F2 P24468 2/20 0.33
RAB9A P51151 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044730 0.93 LMNA (0.39) ALDH1A1ELOVL6TSHRKCNQ1HSD17B10
SCHEMBL4045961 0.93 CTSK (0.39) ALDH1A1ELOVL6TSHRKCNQ1HSD17B10
SCHEMBL4043292 0.91 ALDH1A1 (0.37) ALDH1A1PREPFAPLMNACHRM1
SCHEMBL4044339 0.90 ALDH1A1 (0.37) ALDH1A1PREPFAPLMNANR2F2
SCHEMBL4047431 0.90 ALDH1A1 (0.37) ALDH1A1KMT2APREPFAPNR2F2
SCHEMBL4046799 0.89 ALDH1A1 (0.39) ALDH1A1ELOVL6PREPFAP
SCHEMBL4048312 0.88 KCNQ1 (0.40) ALDH1A1ELOVL6TSHRKCNQ1HSD17B10
SCHEMBL4050093 0.87 HTT (0.41) ALDH1A1ELOVL6TSHRKCNQ1HSD17B10
SCHEMBL4043678 0.86 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2PREPFAPLMNA
SCHEMBL4039771 0.86 ALDH1A1 (0.38) ALDH1A1PREPFAPGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed