SCHEMBL4047478

SCHEMBL4047478

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1)Oc1cccc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.37
MC3R P41968 1/20 0.37
MC1R Q01726 1/20 0.37
CTSK P43235 2/20 0.34
ACE P12821 3/20 0.34
ITGA4 P13612 3/20 0.33
ITGB7 P26010 3/20 0.33
GRIA1 P42261 1/20 0.33
ROCK2 O75116 1/20 0.33
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
F12 P00748 1/20 0.32
TGM2 P21980 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052351 0.92 CNR1 (0.36) MC4RMC3RMC1RCTSKACE
SCHEMBL4041433 0.90 ALDH1A1 (0.35) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL4042676 0.89 CTSB (0.36) MC4RMC3RMC1RCTSKACE
SCHEMBL4044603 0.88 MC4R (0.37) MC4RMC3RMC1RCTSKITGA4
SCHEMBL4042529 0.88 BCL2 (0.38) MC4RMC3RMC1RCTSKACE
SCHEMBL4044768 0.85 CTSL (0.44) CTSKCTSLCTSBCTSS
SCHEMBL6213140 0.84 CTSK (0.44) MC4RMC3RMC1RCTSKACE
SCHEMBL4046533 0.84 MAPK1 (0.36) MC4RMC3RMC1RCTSKACE
SCHEMBL4043465 0.84 MC4R (0.41) MC4RMC3RMC1RCTSKACE
SCHEMBL4040381 0.83 MC4R (0.36) MC4RMC3RMC1RCTSKITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed