SCHEMBL4055

SCHEMBL4055

CN(C)C(CC(Oc1ccc(C(F)(F)F)cc1)C1CCCCC1)OC(=O)C(=O)OC(CC(Oc1ccc(C(F)(F)F)cc1)C1CCCCC1)N(C)C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPT P10636 1/20 0.38
SLC6A9 P48067 5/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ENPP3 O14638 3/20 0.36
ENPP2 Q13822 2/20 0.36
ENPP1 P22413 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3501 0.83 SMN1; SMN2 (0.40) NPC1HPGDRAB9ASMN1; SMN2MAPT
Oxalic Acid SCHEMBL4054 0.77 SLC6A4 (0.50) SLC6A9SLC6A4
Hydrochloric Acid SCHEMBL3937 0.75 SLC6A4 (0.52) HPGDSMN1; SMN2SLC6A9ALDH1A1SLC6A4
SCHEMBL7318201 0.74 SLC6A9 (0.60) NPC1HPGDRAB9ASMN1; SMN2SLC6A9
SCHEMBL4740321 0.73 SLC6A9 (0.57) NPC1RAB9AMAPTSLC6A9ALDH1A1
SCHEMBL3802 0.72 OPRM1 (0.48) NPC1RAB9ASMN1; SMN2SLC6A9PPARG
Oxalic Acid SCHEMBL3500 0.72 MEN1 (0.50) NPC1HPGDRAB9ASMN1; SMN2MAPT
SCHEMBL10539 0.72 SLC7A5 (0.52) NPC1RAB9ASLC6A9PPARGPPARA
SCHEMBL5143084 0.71 SLC6A2 (0.50) SLC6A4SLC6A3
SCHEMBL4660 0.71 HTR1A (0.46) NPC1RAB9ASLC6A9SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5023269-A 3-aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1991-06-11 US disclosed
EP-0273658-B1 3-ARYLOXY-3-SUBSTITUTED PROPANAMINES ELI LILLY AND COMPANY (US) 1990-10-31 EP disclosed
US-4956388-A ANTIDEPRESSANTS, ANTIANXIETY, TREATMENT OF OBESITY, ADDICTION TO SMOKING AND ALCOHOL ELI LILLY AND COMPANY (US) 1990-09-11 US disclosed
EP-0273658-A1 3-Aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed